SCHEMBL8041234

SCHEMBL8041234

COc1cc(Cl)c(C(=O)N(C)C(=O)N2CCOCC2)cc1O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.47
ALDH1A1 P00352 3/20 0.45
KMT2A Q03164 3/20 0.44
MEN1 O00255 1/20 0.44
TRPV1 Q8NER1 1/20 0.43
TSHR P16473 2/20 0.43
FKBP1A P62942 1/20 0.43
HSP90AA1 P07900 1/20 0.42
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA3 P07451 1/20 0.41
CA4 P22748 1/20 0.41
CA6 P23280 1/20 0.41
CA5A P35218 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
CA13 Q8N1Q1 1/20 0.41
CA14 Q9ULX7 1/20 0.41
CA5B Q9Y2D0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8039013 0.88 ALDH1A1 (0.41) POLBALDH1A1KMT2AMEN1TRPV1
SCHEMBL8031648 0.80 SMN1; SMN2 (0.52) ALDH1A1KMT2AMEN1LMNAMAPT
SCHEMBL8035102 0.79 POLB (0.50) POLBALDH1A1KMT2AMEN1TSHR
SCHEMBL8038657 0.76 POLB (0.40) POLBALDH1A1KMT2AMEN1MAPT
SCHEMBL8025473 0.74 HSP90AA1 (0.37) ALDH1A1KMT2AMEN1TSHRHSP90AA1
SCHEMBL8035119 0.74 KDM4E (0.40) ALDH1A1KMT2AMEN1HSP90AA1LMNA
SCHEMBL8039002 0.73 MAPT (0.39) ALDH1A1KMT2AMEN1TSHRHSP90AA1
SCHEMBL8025474 0.72 TSHR (0.39) KMT2AMEN1TSHRHSP90AA1LMNA
SCHEMBL8032092 0.71 ALDH1A1 (0.44) POLBALDH1A1KMT2AMEN1TSHR
SCHEMBL8039016 0.71 HTT (0.42) ALDH1A1TRPV1HSP90AA1LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed