SCHEMBL8043675

SCHEMBL8043675

FC(F)(F)c1cc(-c2csc(Sc3nnnn3-c3cccnc3)n2)cc(C(F)(F)F)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIT P10721 3/20 0.39
HSD17B10 Q99714 1/20 0.38
ABL1 P00519 1/20 0.37
BCR P11274 1/20 0.37
POLB P06746 3/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
HTT P42858 1/20 0.37
TDP1 Q9NUW8 2/20 0.36
GAA P10253 1/20 0.36
KDM4E B2RXH2 1/20 0.35
GRM1 Q13255 2/20 0.35
ALDH1A1 P00352 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
CYP19A1 P11511 1/20 0.34
AXL P30530 1/20 0.34
PBRM1 Q86U86 1/20 0.34
MKNK1 Q9BUB5 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8043200 0.89 ALDH1A1 (0.43) HSD17B10POLBHTTTDP1GAA
SCHEMBL8033936 0.87 ALDH1A1 (0.42) HSD17B10POLBHTTKDM4EALDH1A1
SCHEMBL8044443 0.84 ALDH1A1 (0.49) HSD17B10POLBHTTTDP1KDM4E
SCHEMBL8043905 0.83 KDM4E (0.37) HSD17B10CYP3A4CYP2C19HTTTDP1
SCHEMBL8044564 0.82 CYP19A1 (0.48) HSD17B10POLBCYP3A4CYP2C19HTT
SCHEMBL8050838 0.81 KDM4E (0.36) HSD17B10POLBCYP3A4CYP2C19HTT
SCHEMBL8044497 0.81 HTT (0.33) POLBHTTKDM4EALDH1A1
SCHEMBL8037043 0.81 SMN1; SMN2 (0.39) HSD17B10HTTTDP1GAAKDM4E
SCHEMBL8047017 0.80 HSP90AA1 (0.44) HSD17B10POLBCYP2C9CYP2C19HTT
SCHEMBL8043941 0.80 PTGS2 (0.37) HSD17B10POLBCYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed