SCHEMBL8047017

SCHEMBL8047017

COc1ccc(-n2nnnc2Sc2nc(-c3cc(C(F)(F)F)cc(C(F)(F)F)c3)cs2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.44
HSP90AB1 P08238 1/20 0.44
MAPT P10636 8/20 0.42
ALDH1A1 P00352 6/20 0.42
RAB9A P51151 3/20 0.42
USP2 O75604 3/20 0.42
HPGD P15428 3/20 0.42
GAA P10253 2/20 0.42
SMN1; SMN2 Q16637 5/20 0.41
HTT P42858 3/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
KDM4E B2RXH2 5/20 0.40
LMNA P02545 8/20 0.40
KDM1A O60341 1/20 0.40
TSHR P16473 4/20 0.39
NPSR1 Q6W5P4 2/20 0.39
MAPK1 P28482 1/20 0.39
MEN1 O00255 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8037043 0.89 SMN1; SMN2 (0.39) MAPTALDH1A1RAB9AUSP2HPGD
SCHEMBL8050838 0.87 KDM4E (0.36) MAPTALDH1A1HPGDGAASMN1; SMN2
SCHEMBL8043905 0.87 KDM4E (0.37) MAPTALDH1A1RAB9AUSP2SMN1; SMN2
SCHEMBL8043200 0.87 ALDH1A1 (0.43) MAPTALDH1A1USP2HPGDGAA
SCHEMBL8043941 0.86 PTGS2 (0.37) MAPTALDH1A1RAB9AGAASMN1; SMN2
SCHEMBL8043968 0.83 MEN1 (0.45) ALDH1A1HPGDSMN1; SMN2KDM4ELMNA
SCHEMBL8034319 0.83 ALDH1A1 (0.51) MAPTALDH1A1RAB9AUSP2HPGD
SCHEMBL8033936 0.83 ALDH1A1 (0.42) MAPTALDH1A1HPGDSMN1; SMN2HTT
SCHEMBL8043931 0.83 PTGS2 (0.43) CYP2C9PTGS1PTGS2
SCHEMBL8049946 0.82 ALOX5 (0.47) MAPTALDH1A1RAB9AUSP2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed