SCHEMBL8043690

SCHEMBL8043690

Fc1cccc(F)c1-c1nnc(S)s1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.39
ALDH1A1 P00352 2/20 0.39
PIM1 P11309 3/20 0.34
PIM3 Q86V86 3/20 0.34
PIM2 Q9P1W9 2/20 0.34
SMN1; SMN2 Q16637 3/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA7 P43166 1/20 0.32
CA9 Q16790 1/20 0.32
NPC1 O15118 4/20 0.31
RAB9A P51151 4/20 0.31
RXFP1 Q9HBX9 1/20 0.31
BACE1 P56817 1/20 0.31
MEN1 O00255 1/20 0.31
LMNA P02545 1/20 0.31
PRNP P04156 1/20 0.31
GAA P10253 1/20 0.31
HPGD P15428 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL968101 0.80 KDM4E (0.61) KDM4EALDH1A1PIM1PIM3PIM2
SCHEMBL8047555 0.72 KDM4E (0.65) KDM4EALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL8840237 0.71 TTR (0.43) KDM4EALDH1A1PIM1PIM3SMN1; SMN2
SCHEMBL14557099 0.69 KDM4E (0.43) KDM4EALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL8043829 0.68 KDM4E (0.40) KDM4EALDH1A1PIM1PIM3PIM2
SCHEMBL28353374 0.65 ALDH1A1 (0.48) KDM4EALDH1A1SMN1; SMN2CA1CA2
SCHEMBL11025151 0.64 KDM4E (0.49) KDM4EALDH1A1PIM1PIM3PIM2
SCHEMBL1531740 0.64 PTPN11 (0.47) KDM4EALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL8043317 0.64 HSD17B1 (0.76) SMN1; SMN2RAB9ALMNA
SCHEMBL8042130 0.64 HSD17B1 (0.46) KDM4EALDH1A1SMN1; SMN2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed