SCHEMBL8044714

SCHEMBL8044714

Clc1cnc(Sc2nnn(CCc3ccccc3)n2)s1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.34
ALDH1A1 P00352 4/20 0.34
NPC1 O15118 3/20 0.34
HPGD P15428 3/20 0.34
LMNA P02545 2/20 0.34
KDM4E B2RXH2 1/20 0.34
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
L3MBTL1 Q9Y468 2/20 0.33
MAPT P10636 2/20 0.32
HDAC3 O15379 1/20 0.32
HDAC4 P56524 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC7 Q8WUI4 1/20 0.32
HDAC2 Q92769 1/20 0.32
HDAC10 Q969S8 1/20 0.32
HDAC11 Q96DB2 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8033963 0.89 RAB9A (0.44) RAB9AALDH1A1NPC1HPGDLMNA
SCHEMBL8043417 0.83 HDAC6 (0.36) RAB9ANPC1HPGDLMNAKDM4E
SCHEMBL8042849 0.81 ALDH1A1 (0.33) RAB9AALDH1A1NPC1MAPTSMN1; SMN2
SCHEMBL8032788 0.81 PTGS2 (0.33) KDM4EL3MBTL1KMT2ACYP1A2CYP2C9
SCHEMBL8042797 0.81 MAPK8 (0.43) RAB9AALDH1A1NPC1MAPTHTT
SCHEMBL8046313 0.79 ALDH1A1 (0.35) RAB9AALDH1A1NPC1HPGDLMNA
SCHEMBL8042548 0.78 TRPM8 (0.34) RAB9AALDH1A1NPC1LMNAL3MBTL1
SCHEMBL8042933 0.78 DCUN1D1 (0.37) RAB9AALDH1A1NPC1LMNAKDM4E
SCHEMBL8047827 0.78 NPC1 (0.41) RAB9AALDH1A1NPC1HDAC3HDAC4
SCHEMBL8037025 0.77 MEN1 (0.37) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed