SCHEMBL8043931

SCHEMBL8043931

NS(=O)(=O)c1ccc(-n2nnnc2Sc2nc(-c3cc(C(F)(F)F)cc(C(F)(F)F)c3)cs2)cc1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 15/20 0.43
CYP2C9 P11712 1/20 0.41
PDPK1 O15530 3/20 0.41
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA3 P07451 1/20 0.38
CA4 P22748 1/20 0.38
CA6 P23280 1/20 0.38
CA5A P35218 1/20 0.38
CA7 P43166 1/20 0.38
CA9 Q16790 1/20 0.38
CA13 Q8N1Q1 1/20 0.38
CA14 Q9ULX7 1/20 0.38
CA5B Q9Y2D0 1/20 0.38
PTGS1 P23219 5/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8043905 0.85 KDM4E (0.37)
SCHEMBL8046494 0.85 EP300 (0.42)
SCHEMBL8043200 0.85 ALDH1A1 (0.43)
SCHEMBL8043233 0.84 PTGS2 (0.56) PTGS2CYP2C9CA12CA1CA2
SCHEMBL8043968 0.84 MEN1 (0.45)
SCHEMBL8050838 0.83 KDM4E (0.36) PTGS2PTGS1
SCHEMBL8047017 0.83 HSP90AA1 (0.44) PTGS2CYP2C9PTGS1
SCHEMBL8043941 0.83 PTGS2 (0.37) PTGS2CYP2C9PTGS1
SCHEMBL8050817 0.82 PTGS2 (0.57) PTGS2CA12CA1CA2CA4
SCHEMBL8033936 0.81 ALDH1A1 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed