SCHEMBL8068050

SCHEMBL8068050

CN1CCN(CCCOc2ccc3c(=O)c4[nH]nnc4c(=O)[nH]c3c2)CC1

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
XDH P47989 2/20 0.48
SIGMAR1 Q99720 2/20 0.45
DRD3 P35462 2/20 0.45
HRH3 Q9Y5N1 1/20 0.45
HRH4 Q9H3N8 5/20 0.43
MAOA P21397 1/20 0.42
PARP1 P09874 1/20 0.41
KDM4E B2RXH2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL8067000 0.92 XDH (0.44) XDHSIGMAR1DRD3HRH3HRH4
SCHEMBL7827131 0.92 PARP1 (0.50) XDHSIGMAR1HRH3MAOAPARP1
SCHEMBL8067124 0.90 MAOA (0.52) SIGMAR1HRH3MAOAPARP1KDM4E
SCHEMBL7831263 0.88 ACHE (0.52) HRH3MAOAKDM4E
SCHEMBL8071910 0.84 ACHE (0.53) SIGMAR1HRH3MAOA
Trifluoroacetic Acid SCHEMBL8066735 0.84 MAOA (0.45) SIGMAR1HRH3MAOAPARP1KDM4E
SCHEMBL7826517 0.82 MAOA (0.52) MAOAPARP1KDM4E
SCHEMBL7826175 0.82 MAOA (0.54) SIGMAR1DRD3HRH3MAOAPARP1
SCHEMBL7824605 0.81 CTSV (0.43) MAOA
SCHEMBL7827211 0.81 HSD17B10 (0.51) PARP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6114431-A Plastic composition GRIFFIN CORP. (US) 2000-09-05 US claimed
CN-100558356-C The method that using cyclooxygenase-2-inhibitor 2 treatment and prophylaxis of tumours form G D SIORL & CO (US) 2009-11-11 CN disclosed
CN-1332661-C Methods of treating and preventing neoplasia using cyclooxygenase-2 inhibitors SEARLE & CO (US) 2007-08-22 CN disclosed
CN-1660083-A Method of using benzenesulphoamides that are cyclooxygenase-2-inhibitors in the treatment and prevention of neoplasia G D SIORL & CO (US) 2005-08-31 CN disclosed
US-6093714-A AN ANTIALLERGENS FOR TREATMENT AND PREVENTION OF BRONCHIAL ASTHMA, ECZEMA, HIVES, ALLERGIC GASTROINTESTINAL TROUBLES, ALLERGIC RHINITIS, ALLERGIC CONJUNCTIVITIS MEIJI SEIKA KAISHA, LTD. (JP) 2000-07-25 US disclosed
CN-1247470-A Methods of using cyclooxygenase-2 inhibitors as anti-angiogenic agents SEARLE & CO (US) 2000-03-15 CN disclosed
CN-1244122-A Methods of treating and preventing neoplasia using cyclooxygenase-2 inhibitors SEARLE & CO (US) 2000-02-09 CN disclosed
EP-0422204-A1 PLASTIC CRAYON BINNEY & SMITH INC. (US) 1991-04-17 EP disclosed
WO-1990012845-A1 PLASTIC CRAYON BINNEY & SMITH INC. (US) 1990-11-01 WO disclosed