SCHEMBL8076863

SCHEMBL8076863

COc1ccc2[nH]c(N3CCC(Nc4ccc(C(=O)OC(C)(C)C)cc4)CC3)nc2c1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.50
LMNA P02545 1/20 0.43
POLB P06746 1/20 0.43
MAPT P10636 4/20 0.42
GFER P55789 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
NAMPT P43490 1/20 0.41
FLT3 P36888 1/20 0.41
BACE1 P56817 1/20 0.40
DYRK1A Q13627 1/20 0.40
NPBWR1 P48145 1/20 0.39
NPC1 O15118 1/20 0.39
MAPK1 P28482 1/20 0.39
HTT P42858 1/20 0.39
RAB9A P51151 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
TP53 P04637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8071863 0.88 LMNA (0.47) ALDH1A1LMNAPOLBMAPTGFER
SCHEMBL8071876 0.81 MGLL (0.46) ALDH1A1LMNAPOLBMAPTHTT
SCHEMBL8071618 0.73 DNMT1 (0.45) ALDH1A1MAPTFLT3NPC1MAPK1
SCHEMBL8071641 0.73 ALDH1A1 (0.47) ALDH1A1LMNAPOLBMAPTNPSR1
SCHEMBL8061075 0.73 EHMT2 (0.48) ALDH1A1
SCHEMBL8076826 0.72 ADRA1A (0.56)
SCHEMBL8071878 0.72 GPR119 (0.56) ALDH1A1MAPTNPC1MAPK1HTT
SCHEMBL18428484 0.70 ALDH1A1 (0.59) ALDH1A1MAPTNPSR1NAMPTNPC1
SCHEMBL8071621 0.69 ABCG2 (0.48) ALDH1A1LMNAMAPTNPSR1NPC1
SCHEMBL4243494 0.69 ALDH1A1 (0.76) ALDH1A1MAPTNPSR1NPC1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6156758-A Antibacterial quinazoline compounds ISIS PHARMACEUTICALS, INC. (US) 2000-12-05 US disclosed