SCHEMBL8090158

SCHEMBL8090158

CNC(=O)Nc1ccc(-c2nc(N)cc(C3(S(=O)(=O)c4ccc(Cl)cc4)CCOCC3)n2)cc1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MTOR P42345 9/20 0.46
PIK3CA P42336 7/20 0.46
PIK3CG P48736 5/20 0.46
PIK3CD O00329 8/20 0.42
ALDH1A1 P00352 1/20 0.40
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8083160 0.88 PIK3CD (0.43) MTORPIK3CAPIK3CGPIK3CDCA12
SCHEMBL8093573 0.87 PIK3CA (0.46) MTORPIK3CAPIK3CGPIK3CD
SCHEMBL8092043 0.86 MTOR (0.49) MTORPIK3CAPIK3CGPIK3CD
SCHEMBL8092637 0.86 KMT2A (0.42) MTORPIK3CAPIK3CGPIK3CDCA12
SCHEMBL8097257 0.86 ALDH1A1 (0.41) MTORPIK3CAPIK3CGALDH1A1CA12
SCHEMBL8083973 0.85 ALDH1A1 (0.43) MTORPIK3CAPIK3CGPIK3CDALDH1A1
SCHEMBL8090246 0.85 PIK3CA (0.42) MTORPIK3CAPIK3CGPIK3CDALDH1A1
SCHEMBL8094423 0.84 CA2 (0.43) MTORPIK3CAPIK3CGALDH1A1CA12
SCHEMBL8083874 0.84 MTOR (0.47) MTORPIK3CAPIK3CGPIK3CD
SCHEMBL8099749 0.84 MTOR (0.40) MTORPIK3CAPIK3CGPIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed