SCHEMBL8098096

SCHEMBL8098096

N=C(N)NCCC[C@H](NC=O)OB(O)C1(C(=O)NCCc2ccc3ccccc3c2)CCCC1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.35
MAPT P10636 4/20 0.33
HTT P42858 3/20 0.33
LMNA P02545 1/20 0.33
MC3R P41968 2/20 0.33
MC1R Q01726 2/20 0.33
MC4R P32245 1/20 0.33
RXFP1 Q9HBX9 1/20 0.32
FURIN P09958 1/20 0.31
TGM2 P21980 1/20 0.31
NAMPT P43490 1/20 0.31
TSHR P16473 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
SLC1A3 P43003 1/20 0.31
SLC1A2 P43004 1/20 0.31
SLC1A1 P43005 1/20 0.31
GRB2 P62993 1/20 0.30
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8098063 0.90 CES2 (0.37) CES2MAPTHTTLMNAMC3R
SCHEMBL8091511 0.87 SMN1; SMN2 (0.40) LMNANAMPTSMN1; SMN2ALDH1A1POLB
SCHEMBL8090119 0.81 CAPN1 (0.33) LMNASMN1; SMN2KDM4EALDH1A1PKM
SCHEMBL8091691 0.79 ALDH1A1 (0.33) TSHRALDH1A1
SCHEMBL8083619 0.78 SMN1; SMN2 (0.42) LMNASMN1; SMN2ALDH1A1POLB
SCHEMBL8096021 0.71 CYP1A2 (0.37) CES2MAPTHTTLMNAMC3R
SCHEMBL8090174 0.67 F2 (0.39) KDM4ECYP1A2
SCHEMBL8095300 0.67 CYP3A4 (0.36) TSHRALDH1A1CYP1A2
SCHEMBL8090189 0.66 MMP8 (0.37) KDM4ECYP1A2
SCHEMBL21171990 0.66 HDAC1 (0.50) MC3RMC1RMC4RCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0792883-B1 Novel derivates of boronic acid, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 2000-12-20 EP disclosed
EP-0792883-A1 Novel derivates of boronic acid, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1997-09-03 EP disclosed