SCHEMBL8101320

SCHEMBL8101320

CN(C)CCCN1c2cccnc2N(CCCN(C)C)c2nc([N+](=O)[O-])ccc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 4/20 0.40
LMNA P02545 4/20 0.40
ALDH1A1 P00352 4/20 0.40
CHRM2 P08172 3/20 0.40
HTR1A P08908 3/20 0.40
DRD1 P21728 3/20 0.40
SLC6A4 P31645 3/20 0.40
DRD3 P35462 3/20 0.40
MAPT P10636 3/20 0.40
CYP1A2 P05177 3/20 0.40
SLC22A1 O15245 2/20 0.40
PRNP P04156 2/20 0.40
CHRM4 P08173 2/20 0.40
CHRM5 P08912 2/20 0.40
CHRM1 P11229 2/20 0.40
DRD2 P14416 2/20 0.40
ADRA2B P18089 2/20 0.40
ADRA2C P18825 2/20 0.40
CHRM3 P20309 2/20 0.40
DRD4 P21917 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8101312 0.97 HTR1A (0.39) CYP2D6LMNAALDH1A1CHRM2HTR1A
SCHEMBL8103181 0.91 ALDH1A1 (0.42) CYP2D6LMNAALDH1A1CHRM2HTR1A
SCHEMBL8101460 0.87 PKM (0.36) ALDH1A1MAPTCYP1A2TP53CYP2C19
SCHEMBL8093559 0.87 ALDH1A1 (0.43) CYP2D6LMNAALDH1A1CHRM2HTR1A
SCHEMBL8107634 0.84 PKM (0.37) LMNAALDH1A1MAPTCYP1A2TP53
SCHEMBL8101555 0.83 CYP2D6 (0.54) CYP2D6LMNAALDH1A1CHRM2HTR1A
SCHEMBL8103445 0.80 CYP2D6 (0.44) CYP2D6LMNAALDH1A1CHRM2HTR1A
SCHEMBL8093557 0.79 CYP2D6 (0.51) CYP2D6LMNAALDH1A1CHRM2HTR1A
SCHEMBL8103441 0.77 KDM4E (0.38) LMNAALDH1A1MAPTCYP1A2TP53
SCHEMBL8107912 0.76 CYP2D6 (0.42) CYP2D6LMNAALDH1A1CHRM2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6127369-A 5,10-dihydrodipyrido[2,3-b:2,3-e]pyrazin and 5,10-dihydrodipyrido[2,3-b:3,2-e]pyrazin compounds ADIR ET COMPAGNIE (FR) 2000-10-03 US disclosed