SCHEMBL8111908

SCHEMBL8111908

CCOC(=O)C(CC)(C(=O)O)C(c1ccccc1)c1ccccc1Cl

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 1/20 0.48
PIN1 Q13526 1/20 0.39
ALDH1A1 P00352 4/20 0.38
TSHR P16473 2/20 0.38
MMP8 P22894 1/20 0.37
ACP3 P15309 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.36
CYP1A2 P05177 3/20 0.36
CYP3A4 P08684 3/20 0.36
CYP2C9 P11712 3/20 0.36
CYP2C19 P33261 3/20 0.36
CYP2D6 P10635 2/20 0.36
HPGD P15428 2/20 0.36
MDM4 O15151 1/20 0.36
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36
MDM2 Q00987 1/20 0.36
IDO1 P14902 1/20 0.35
TDO2 P48775 1/20 0.35
IDO2 Q6ZQW0 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5679986 0.72 CASP1 (0.56) CASP1PIN1ALDH1A1TSHRMMP8
SCHEMBL7109215 0.71 NPC1 (0.52) PIN1ALDH1A1TSHRMMP8SMN1; SMN2
SCHEMBL6076118 0.70 PIN1 (0.44) CASP1PIN1ALDH1A1TSHRMMP8
SCHEMBL578529 0.70 ALDH1A1 (0.56) PIN1ALDH1A1TSHRMMP8CYP1A2
SCHEMBL27774182 0.69 MMP8 (0.44) PIN1ALDH1A1TSHRMMP8SMN1; SMN2
SCHEMBL11069746 0.69 PIN1 (0.49) PIN1ALDH1A1TSHRMMP8SMN1; SMN2
SCHEMBL8998830 0.69 PIN1 (0.45) PIN1ALDH1A1TSHRMMP8MDM4
SCHEMBL5861445 0.69 CASP1 (0.59) CASP1PIN1ALDH1A1TSHRMMP8
SCHEMBL8102772 0.69 CASP1 (0.49) CASP1TSHRMMP8ACP3SMN1; SMN2
SCHEMBL4632797 0.68 CASP1 (0.70) CASP1PIN1ALDH1A1TSHRMMP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0645378-B1 Condensed seven- or eight-membered heterocyclic compounds useful as squalene synthetase inhibitors TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2000-08-23 EP disclosed
US-5698691-A ANTICHOLESTEROL AGENT; SYNTHETASE INHIBITOR; FUNGICIDE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-12-16 US disclosed
EP-0645378-A1 Condensed seven- or eight-membered heterocyclic compounds useful as squalene synthetase inhibitors Takeda Chemical Industries, Ltd. (JP) 1995-03-29 EP disclosed