SCHEMBL8150877

SCHEMBL8150877

N#Cc1ccc(C(c2c[nH]cn2)C(c2ccccc2)(c2ccccc2)c2ccccc2)cc1OCC(F)(F)F

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.35
SLC6A2 P23975 2/20 0.35
SLC6A4 P31645 2/20 0.35
NOS2 P35228 2/20 0.35
S1PR1 P21453 2/20 0.31
AR P10275 4/20 0.30
CTSS P25774 1/20 0.30
SCN9A Q15858 1/20 0.30
S1PR3 Q99500 1/20 0.30
S1PR5 Q9H228 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8155536 0.86 IMPDH2 (0.36) S1PR1ARSCN9AS1PR3
SCHEMBL8149150 0.83 NR3C1 (0.35) S1PR1S1PR3
SCHEMBL7677950 0.82 CYP11B1 (0.36) S1PR1S1PR3
SCHEMBL8155413 0.79 ALDH1A1 (0.36)
SCHEMBL8157364 0.77 XDH (0.36)
SCHEMBL5891827 0.75 CYP19A1 (0.36)
SCHEMBL7669882 0.74 VNN1 (0.35) SLC6A2SLC6A4
SCHEMBL18119750 0.70 AR (0.40) CYP2D6SLC6A2SLC6A4NOS2AR
SCHEMBL7663652 0.69
SCHEMBL7675183 0.68 KIF11 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6077853-A Inhibitors of farnesyl-protein transferase MERCK & CO., INC. (US) 2000-06-20 US disclosed
US-5939439-A Inhibitors of farnesyl-protein transferase MERCK & CO., INC. (US) 1999-08-17 US disclosed