SCHEMBL8228786

SCHEMBL8228786

CC(C)Cn1c(-c2ccccc2)nc2ccccc21

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.67
SMN1; SMN2 Q16637 1/20 0.67
HSD17B10 Q99714 3/20 0.64
LMNA P02545 3/20 0.64
TSHR P16473 1/20 0.64
KDM4E B2RXH2 7/20 0.63
HPGD P15428 3/20 0.63
PDE6D O43924 1/20 0.62
ALDH2 P05091 1/20 0.62
ALDH3A1 P30838 1/20 0.62
TP53 P04637 4/20 0.60
PRKACA P17612 1/20 0.59
RPS6KB1 P23443 1/20 0.59
GSK3B P49841 1/20 0.59
ROCK1 Q13464 1/20 0.59
GAA P10253 2/20 0.57
NPC1 O15118 1/20 0.57
GLA P06280 1/20 0.57
HTT P42858 1/20 0.57
RAB9A P51151 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13784140 0.90 HSD17B10 (0.58) ALDH1A1SMN1; SMN2HSD17B10LMNATSHR
SCHEMBL31267426 0.88 KDM4E (0.72) ALDH1A1SMN1; SMN2HSD17B10LMNATSHR
SCHEMBL22819342 0.86 KDM4E (0.73) ALDH1A1SMN1; SMN2HSD17B10LMNATSHR
SCHEMBL13299519 0.85 NLRP3 (0.72) ALDH1A1SMN1; SMN2HSD17B10LMNATSHR
SCHEMBL12145817 0.83 KDM4E (0.67) ALDH1A1SMN1; SMN2HSD17B10LMNATSHR
SCHEMBL13451619 0.83 KDM4E (0.62) ALDH1A1SMN1; SMN2HSD17B10LMNATSHR
SCHEMBL31267379 0.82 ALDH1A1 (0.64) ALDH1A1SMN1; SMN2HSD17B10LMNAKDM4E
SCHEMBL13127436 0.81 LMNA (0.73) ALDH1A1SMN1; SMN2LMNATSHRKDM4E
SCHEMBL5009162 0.81 KDM4E (0.77) ALDH1A1SMN1; SMN2HSD17B10LMNATSHR
SCHEMBL15314761 0.80 KDM4E (0.58) ALDH1A1HSD17B10LMNATSHRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8501786-B2 Hydroxymethyl pyrrolidines as beta 3 adrenergic receptor agonists MERCK SHARP & DOHME CORP. (US) 2013-08-06 US disclosed
US-8367223-B2 Heteroleptic phosphorescent emitters UNIVERSAL DISPLAY CORPORATION (US) 2013-02-05 US disclosed
US-8367223-B2 Heteroleptic phosphorescent emitters UNIVERSAL DISPLAY CORPORATION (US) 2013-02-05 US disclosed
US-20110028461-A1 HYDROXYMETHYL PYRROLIDINES AS BETA 3 ADRENERGIC RECEPTOR AGONISTS MERCK SHARP & DOHME LLC 2011-02-03 US disclosed
US-20100144591-A1 BENZIMIDAZOLE DERIVATIVES AND METHODS OF USE THEREOF SCHERING CORPORATION 2010-06-10 US disclosed
US-20100141127-A1 PHOSPHORESCENT EMITTERS UNIVERSAL DISPLAY CORPORATION (US) 2010-06-10 US disclosed
US-20100141127-A1 PHOSPHORESCENT EMITTERS UNIVERSAL DISPLAY CORPORATION (US) 2010-06-10 US disclosed
WO-2010056669-A1 PHOSPHORESCENT EMITTERS UNIVERSAL DISPLAY CORPORATION (US) 2010-05-20 WO disclosed
US-20070142369-A1 Combination of an H3 antagonist/inverse agonist and an appetite suppressant SCHERING CORPORATION 2007-06-21 US disclosed
US-20070142369-A1 Combination of an H3 antagonist/inverse agonist and an appetite suppressant SCHERING CORPORATION 2007-06-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070142369-A1 Combination of an H3 antagonist/inverse agonist and an appetite suppressant CNR2, GPR119, GLP1R ALDH1A1 3184/4885SMN1; SMN2 4298/4885HSD17B10 525/4885
US-20100141127-A1 PHOSPHORESCENT EMITTERS PAICS, TYMP, NUDT1 ALDH1A1 695/4885SMN1; SMN2 3461/4885HSD17B10 4746/4885
US-20110028461-A1 HYDROXYMETHYL PYRROLIDINES AS BETA 3 ADRENERGIC RECEPTOR AGONISTS ADRB3, ADRB1, ADRB2 ALDH1A1 352/4885SMN1; SMN2 3396/4885HSD17B10 1355/4885
US-20100144591-A1 BENZIMIDAZOLE DERIVATIVES AND METHODS OF USE THEREOF GPR119, GK, GCK ALDH1A1 612/4885SMN1; SMN2 1534/4885HSD17B10 936/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.