SCHEMBL8299304

SCHEMBL8299304

CC(C)(C)OC(=O)N[C@H](C(=O)O)C12CC3CC(CC(C3)C1)C2

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.48
MEN1 O00255 3/20 0.48
MAPK1 P28482 1/20 0.48
HDAC4 P56524 1/20 0.44
HDAC1 Q13547 1/20 0.44
ALDH1A1 P00352 3/20 0.43
NPC1 O15118 1/20 0.41
EPHX2 P34913 2/20 0.39
GAA P10253 1/20 0.39
CACNA1H O95180 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
CTSS P25774 1/20 0.36
CTSK P43235 1/20 0.36
ALOX15 P16050 1/20 0.36
ITGB3 P05106 1/20 0.36
ITGA2B P08514 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA7 P43166 1/20 0.36
BTK Q06187 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27978333 1.00 KMT2A (0.48) KMT2AMEN1MAPK1HDAC4HDAC1
SCHEMBL15535916 1.00 KMT2A (0.48) KMT2AMEN1MAPK1HDAC4HDAC1
SCHEMBL30170170 0.94 KMT2A (0.41) KMT2AMEN1MAPK1HDAC4HDAC1
SCHEMBL18631592 0.94 KMT2A (0.41) KMT2AMEN1MAPK1HDAC4HDAC1
SCHEMBL24815908 0.86 KMT2A (0.39) KMT2AMEN1MAPK1HDAC4HDAC1
SCHEMBL2110140 0.86 KMT2A (0.39) KMT2AMEN1MAPK1HDAC4HDAC1
SCHEMBL2549745 0.86 KMT2A (0.39) KMT2AMEN1MAPK1HDAC4HDAC1
SCHEMBL27218008 0.86 KMT2A (0.39) KMT2AMEN1MAPK1HDAC4HDAC1
SCHEMBL8271718 0.86 KMT2A (0.39) KMT2AMEN1MAPK1HDAC4HDAC1
SCHEMBL27218038 0.86 KMT2A (0.39) KMT2AMEN1MAPK1HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 32 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3759075-B1 COMPOUNDS WITH FERROPTOSIS INDUCING ACTIVITY AND METHODS OF THEIR USE FERRO THERAPEUTICS INC (US) 2025-07-23 EP disclosed
WO-2025090919-A1 COMPOSITIONS AND METHODS FOR TREATING INFLAMMATORY BOWEL DISEASE PITON THERAPEUTICS, INC. (US) 2025-05-01 WO disclosed
WO-2025090920-A1 COMPOSITIONS AND METHODS FOR TREATING DYSFUNCTION OF GLUCOSE METABOLISM AND/OR REGULATION PITON THERAPEUTICS, INC. (US) 2025-05-01 WO disclosed
US-20240197666-A1 DITERPENOID COMPOUNDS THAT ACT ON PROTEIN KINASE C (PKC) K-GEN THERAPEUTICS, INC. (US) 2024-06-20 US disclosed
EP-4313095-A1 DITERPENOID COMPOUNDS THAT ACT ON PROTEIN KINASE C (PKC) K-Gen Therapeutics, Inc. (US) 2024-02-07 EP disclosed
US-20230372372-A1 COMBINATION THERAPIES USING CASPASE-1 DEPENDENT ANTICANCER AGENTS AND PGE2 ANTAGONISTS TRUSTEES OF TUFTS COLLEGE 2023-11-23 US disclosed
CN-117098544-A Diterpenoid compounds acting on Protein Kinase C (PKC) K-GEN治疗股份有限公司 2023-11-21 CN disclosed
US-20230312571-A1 RING-MODIFIED PROLINE SHORT PEPTIDE COMPOUND AND USE THEREOF FUJIAN AKEYLINK BIOTECHNOLOGY CO., LTD. (CN) 2023-10-05 US disclosed
EP-4209494-A1 RING-MODIFIED PROLINE SHORT PEPTIDE COMPOUND AND USE THEREOF Fujian Akeylink Biotechnology Co., Ltd. (CN) 2023-07-12 EP disclosed
US-11583516-B2 Dash inhibitors, and uses related thereto TRUSTEES OF TUFTS COLLEGE (US) 2023-02-21 US disclosed
US-20190209525-A1 DASH INHIBITORS, AND USES RELATED THERETO TRUSTEES OF TUFTS COLLEGE 2019-07-11 US disclosed
EP-2995615-A1 CYCLOPROPYL-FUSED PYRROLIDINE-BASED INHIBITORS OF DIPEPTIDYL PEPTIDASE IV AND THEIR PHARMACEUTICAL USE AstraZeneca AB (SE) 2016-03-16 EP disclosed
WO-2014118612-A1 PROCESS FOR THE PREPARATION OF INTERMEDIATES OF SYNTHESIS OF SAXAGLIPTIN AND NOVEL COMPOUNDS LABORATORIO CHIMICO INTERNAZIONALE S.P.A. (IT) 2014-08-07 WO disclosed
WO-2013175395-A2 IMPROVED PROCESS FOR PREPARATION OF SAXAGLIPTIN AND ITS SALTS DR. REDDYS LABORATORIES LIMITED (IN) 2013-11-28 WO disclosed
WO-2013111158-A2 PROCESS FOR THE PREPARATION OF DPP-IV INHIBITOR MSN LABORATORIES LIMITED (IN) 2013-08-01 WO disclosed
US-RE44186-E1 Cyclopropyl-fused pyrrolidine-based inhibitors of dipeptidyl peptidase IV and method BRISTOL-MYERS SQUIBB COMPANY (US) 2013-04-30 US disclosed
EP-2272825-A2 N-Protected amino hydroxy adamantane carboxylic acid and process for its preparation Bristol-Myers Squibb Company (US) 2011-01-12 EP disclosed
EP-1553937-B1 GLYCINENITRILE-BASED INHIBITORS OF DIPEPTIDYL PEPTIDASE IV BRISTOL MYERS SQUIBB CO (US) 2010-06-02 EP disclosed
WO-2005012249-A2 ADAMANTYGLYCINE- BASED INHIBITORS OF DIPEPTIDYL PEPTIDASE IV FOR THE TREATMENT OF DIABETES BRISTOL-MYERS SQUIBB COMPANY (US) 2005-02-10 WO disclosed
WO-2004037181-A2 GLYCINENITRILE-BASED INHIBITORS OF DIPEPTIDYL PEPTIDASE IV AND METHODS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-05-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11583516-B2 Dash inhibitors, and uses related thereto PCNA, CD2BP2, CCNO KMT2A 1719/4885MEN1 2512/4885MAPK1 1154/4885
US-20230372372-A1 COMBINATION THERAPIES USING CASPASE-1 DEPENDENT ANTICANCER AGENTS AND PGE2 ANTAGONISTS CASP1, CASP2, APAF1 KMT2A 3963/4885MEN1 3338/4885MAPK1 1034/4885
US-20230312571-A1 RING-MODIFIED PROLINE SHORT PEPTIDE COMPOUND AND USE THEREOF VIP, PREP, PRAP1 KMT2A 3623/4885MEN1 1707/4885MAPK1 998/4885
US-20190209525-A1 DASH INHIBITORS, AND USES RELATED THERETO CD2BP2, PCNA, CD2 KMT2A 1488/4885MEN1 2401/4885MAPK1 1172/4885
US-20240197666-A1 DITERPENOID COMPOUNDS THAT ACT ON PROTEIN KINASE C (PKC) PRKCA, PRKCB, PRKCI KMT2A 3236/4885MEN1 4010/4885MAPK1 300/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.