SCHEMBL8302093

SCHEMBL8302093

CC(C)(Cc1ccsc1)CN1CCN(c2cccc3c2CCOO3)CC1

nearest known ligand 0.39

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.39
HTR1A P08908 2/20 0.33
DRD2 P14416 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8306494 0.84 ALDH1A1 (0.52) ALDH1A1HTR1ADRD2
SCHEMBL8303869 0.83 ALDH1A1 (0.40) ALDH1A1HTR1ADRD2
SCHEMBL8303199 0.81 HTR1A (0.43) ALDH1A1HTR1ADRD2
SCHEMBL8303555 0.80 HTR1A (0.47) ALDH1A1HTR1ADRD2
SCHEMBL8304635 0.70 DRD4 (0.43) ALDH1A1HTR1ADRD2
SCHEMBL8303443 0.68 HTR1A (0.58) HTR1ADRD2
SCHEMBL9179387 0.67 SIGMAR1 (0.53) ALDH1A1HTR1ADRD2
SCHEMBL8691571 0.66 MTNR1A (0.36)
SCHEMBL6193067 0.66 ADRB1 (0.54) ALDH1A1HTR1ADRD2
SCHEMBL8306501 0.66 HTR1A (0.63) ALDH1A1HTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0574313-B1 1,4-Disubstituted piperazines for the treatment of disorders of the central nervous system and neuro-endocrine disorders ADIR (FR) 1999-10-06 EP disclosed
US-5464834-A Antidepressants, central nervous system ADIR ET COMPAGNIE (FR) 1995-11-07 US disclosed
EP-0574313-A1 1,4-Disubstituted piperazines for the treatment of disorders of the central nervous system and neuro-endocrine disorders ADIR ET COMPAGNIE (FR) 1993-12-15 EP disclosed