SCHEMBL8302750

SCHEMBL8302750

CCc1cccc(CC)c1N(C)C(=O)c1ccc([N+](=O)[O-])c([N+](=O)[O-])c1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CASP6 P55212 1/20 0.48
PDK1 Q15118 1/20 0.45
SMN1; SMN2 Q16637 4/20 0.44
ALDH1A1 P00352 4/20 0.44
HCAR3 P49019 5/20 0.42
KMT2A Q03164 4/20 0.40
LMNA P02545 2/20 0.40
ATM Q13315 1/20 0.40
MAPT P10636 3/20 0.39
HTT P42858 2/20 0.39
MEN1 O00255 2/20 0.39
NPC1 O15118 1/20 0.39
MAPK1 P28482 1/20 0.39
RAB9A P51151 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8304450 0.86 CASP6 (0.47) CASP6PDK1SMN1; SMN2ALDH1A1HCAR3
SCHEMBL8305734 0.81 PDK1 (0.47) CASP6PDK1SMN1; SMN2ALDH1A1HCAR3
SCHEMBL8303776 0.78 ATM (0.65) CASP6SMN1; SMN2ALDH1A1HCAR3KMT2A
SCHEMBL9188252 0.76 CASP6 (0.57) CASP6SMN1; SMN2ALDH1A1HCAR3LMNA
SCHEMBL8300884 0.75 CASP6 (0.49) CASP6SMN1; SMN2ALDH1A1HCAR3KMT2A
SCHEMBL8307952 0.75 ALDH1A1 (0.57) CASP6PDK1SMN1; SMN2ALDH1A1HCAR3
SCHEMBL5913206 0.75 PDK1 (0.62) CASP6PDK1SMN1; SMN2ALDH1A1HCAR3
SCHEMBL8306708 0.74 PDK1 (0.48) CASP6PDK1ALDH1A1KMT2AMAPT
SCHEMBL8305961 0.74 ALDH1A1 (0.50) CASP6SMN1; SMN2ALDH1A1HCAR3KMT2A
SCHEMBL8302742 0.73 ALDH1A1 (0.50) CASP6PDK1SMN1; SMN2ALDH1A1HCAR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934068-A1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 1999-08-11 EP claimed
WO-1998009630-A1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 1998-03-12 WO claimed
EP-0934068-A1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 1999-08-11 EP disclosed
WO-1998009630-A1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 1998-03-12 WO disclosed