SCHEMBL8309008

SCHEMBL8309008

CC(=NO)c1ccc(-c2ccc(C(F)(F)F)cc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 6/20 0.50
CES2 O00748 1/20 0.45
CES1 P23141 1/20 0.45
NR4A1 P22736 1/20 0.43
NR4A2 P43354 1/20 0.43
NR4A3 Q92570 1/20 0.43
S1PR1 P21453 1/20 0.41
PTGS1 P23219 2/20 0.41
NQO2 P16083 1/20 0.41
PTGS2 P35354 1/20 0.41
RXRA P19793 1/20 0.41
RXRB P28702 1/20 0.41
RXRG P48443 1/20 0.41
MTOR P42345 2/20 0.40
CA9 Q16790 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL266456 0.94 CES2 (0.50) CES2CES1NR4A1NR4A2NR4A3
SCHEMBL4022029 0.94 CES2 (0.50) CES2CES1NR4A1NR4A2NR4A3
SCHEMBL13645704 0.83 CA9 (0.47) CA9ALDH1A1LMNARAB9A
Trifluoromethylbenzene SCHEMBL28068069 0.81 ALDH1A1 (0.54) KIF11CES2NR4A1NR4A2NR4A3
SCHEMBL5609938 0.78 LMNA (0.50) CES2CES1CA9ALDH1A1LMNA
SCHEMBL6377926 0.77 MMP2 (0.45) KIF11RAB9A
SCHEMBL17574261 0.76 CES2 (0.48) CES2CES1NR4A1NR4A2NR4A3
SCHEMBL4835788 0.76 CES2 (0.59) KIF11CES2CES1NR4A1NR4A2
SCHEMBL8308938 0.76 CYP17A1 (0.46) KIF11CA9LMNA
SCHEMBL28127817 0.76 CES2 (0.48) CES2CES1NR4A1NR4A2NR4A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5972959-A Oxime derivatives, their preparation and their therapeutic use SANKYO COMPANY, LIMITED (JP) 1999-10-26 US disclosed
EP-0708098-B1 Oxime derivatives, their preparation and their therapeutic use SANKYO CO (JP) 1999-03-03 EP disclosed
US-5780490-A A O-(2,4-OXA(OR THIA)ZOLIDINYL)PHENYLOXY(OR THIO OR AMINO) ALKYLOXIME; ALDOSE REDUCTASE INHIBITORS; ANTIDIABETIC AND -HYPOGLYCEMIC AGENTS; LIVER, SKIN AND UROGENITAL DISORDERS SANKYO COMPANY, LIMITED (JP) 1998-07-14 US disclosed
US-5703096-A ANTIDIABETIC AGENTS; ALDOSE REDUCTASE INHIBITOR SANKYO COMPANY, LIMITED (JP) 1997-12-30 US disclosed
EP-0708098-A1 Oxime derivatives, their preparation and their therapeutic use SANKYO COMPANY LIMITED (JP) 1996-04-24 EP disclosed