SCHEMBL8323488

SCHEMBL8323488

CC(N)([CH]c1ccc(F)c(Cl)c1)Cc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 3/20 0.41
TAAR1 Q96RJ0 1/20 0.41
TRPA1 O75762 1/20 0.36
SLC6A4 P31645 2/20 0.36
SLC6A3 Q01959 2/20 0.36
HTR2A P28223 1/20 0.36
HRH1 P35367 1/20 0.36
HTR2B P41595 1/20 0.36
CHRNA4 P43681 1/20 0.36
KIF11 P52732 4/20 0.33
PTGES O14684 1/20 0.33
G6PC1 P35575 1/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2B Q13224 1/20 0.33
EGFR P00533 1/20 0.33
PTGS2 P35354 2/20 0.33
CYP2D6 P10635 2/20 0.33
CYP3A4 P08684 1/20 0.33
KCNH2 Q12809 1/20 0.33
MEN1 O00255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8323030 0.81 SLC6A2 (0.44) SLC6A2TAAR1SLC6A4SLC6A3HTR2A
SCHEMBL8321757 0.79 SLC6A2 (0.48) SLC6A2TAAR1TRPA1KIF11GRIN1
SCHEMBL8325974 0.78 NFE2L2 (0.46) SLC6A2TAAR1CYP2D6CYP3A4MAPT
SCHEMBL8323216 0.77 SLC6A2 (0.46) SLC6A2TAAR1SLC6A4SLC6A3HTR2A
SCHEMBL8324902 0.75 MAOB (0.49) SLC6A2TAAR1TRPA1CYP2D6CYP3A4
SCHEMBL8323792 0.74 SLC6A2 (0.50) SLC6A2TAAR1TRPA1KIF11CYP2D6
SCHEMBL8323288 0.74 TAAR1 (0.46) SLC6A2TAAR1KIF11GRIN1GRIN2B
SCHEMBL8324690 0.74 TAAR1 (0.46) SLC6A2TAAR1CYP2D6LMNA
SCHEMBL8321777 0.73 GRIN1 (0.45) SLC6A2TAAR1HTR2AHTR2BGRIN1
SCHEMBL8327003 0.71 TRPA1 (0.38) SLC6A2TAAR1TRPA1SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0948496-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDONE COMPOUNDS AND METHODS OF USE Amgen inc. (US) 1999-10-13 EP disclosed
WO-1998024780-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDINONE COMPOUNDS AND THEIR USE AMGEN INC. (US) 1998-06-11 WO disclosed