SCHEMBL8325346

SCHEMBL8325346

COC(CNCc1ccc(F)cc1)CNc1c(C#N)c(=N)n(C)c(=S)n1C

nearest known ligand 0.33

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.33
KDM4E B2RXH2 1/20 0.33
POLB P06746 1/20 0.33
GAA P10253 1/20 0.33
LMNA P02545 2/20 0.33
L3MBTL1 Q9Y468 2/20 0.32
TDP1 Q9NUW8 1/20 0.32
MITF O75030 1/20 0.32
CNR1 P21554 1/20 0.32
CNR2 P34972 1/20 0.32
GPR35 Q9HC97 1/20 0.32
GPR55 Q9Y2T6 1/20 0.32
XBP1 P17861 1/20 0.32
MAPK1 P28482 1/20 0.32
HTT P42858 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
NPC1 O15118 1/20 0.31
GRM5 P41594 1/20 0.31
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8328279 0.86 DNM1 (0.39) ALDH1A1KDM4EPOLBGAALMNA
SCHEMBL8322051 0.83 ALDH1A1 (0.42) ALDH1A1KDM4EPOLBGAAL3MBTL1
SCHEMBL8324185 0.81 CHRM2 (0.39) ALDH1A1KDM4EPOLBGAALMNA
SCHEMBL8328869 0.81 CHRM2 (0.44) ALDH1A1KDM4EPOLBGAALMNA
SCHEMBL8329010 0.81 CHRM2 (0.41) ALDH1A1KDM4EPOLBGAALMNA
SCHEMBL8330575 0.80 MEN1 (0.35) ALDH1A1KDM4EPOLBGAALMNA
SCHEMBL8325662 0.80 CHRM2 (0.46) ALDH1A1KDM4EPOLBGAALMNA
SCHEMBL8328033 0.77 CTSS (0.32)
SCHEMBL8329466 0.73 NRP1 (0.33) ALDH1A1KDM4EGAAL3MBTL1MAPK1
SCHEMBL8324755 0.71 SIGMAR1 (0.37) ALDH1A1GAAMITFMAPK1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0760368-B1 PYRIMIDINE DERIVATIVES NISSHIN FLOUR MILLING CO (JP) 1999-07-28 EP disclosed
US-5736550-A TREATMENT OF GASTROINTESTINAL TRACT DISORDERS NISSHIN FLOUR MILLING CO., LTD. (JP) 1998-04-07 US disclosed
EP-0760368-A1 NOVEL PYRIMIDINE DERIVATIVE NISSHIN FLOUR MILLING CO., LTD. (JP) 1997-03-05 EP disclosed