SCHEMBL8334114

SCHEMBL8334114

CCCC(=O)N(C)C1C(c2cccc(OC)c2)C1(F)F

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SLC9A1 P19634 1/20 0.41
MTNR1B P49286 8/20 0.40
MTNR1A P48039 7/20 0.40
CACNA1D Q01668 1/20 0.39
TSHR P16473 1/20 0.39
KDM1A O60341 1/20 0.38
RCOR1 Q9UKL0 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8333365 0.87 SLC9A1 (0.47) SLC9A1MTNR1BMTNR1ATSHRKDM1A
SCHEMBL8334052 0.81 SLC9A1 (0.43) SLC9A1MTNR1BMTNR1ACACNA1DTSHR
SCHEMBL8329351 0.76 HTR2A (0.47) SLC9A1MTNR1BMTNR1A
SCHEMBL8332882 0.76 HTR2A (0.47) SLC9A1MTNR1BMTNR1A
SCHEMBL8103541 0.76 MTNR1B (0.50) MTNR1BMTNR1A
SCHEMBL8103536 0.76 MTNR1B (0.50) MTNR1BMTNR1A
SCHEMBL28746510 0.69 MTNR1A (0.57) MTNR1BMTNR1A
SCHEMBL8333438 0.69 SLC9A1 (0.39) SLC9A1MTNR1BMTNR1AKDM1ARCOR1
SCHEMBL8333441 0.69 SLC9A1 (0.39) SLC9A1MTNR1BMTNR1AKDM1ARCOR1
SCHEMBL8330356 0.68 SLC9A1 (0.44) SLC9A1MTNR1BMTNR1ACACNA1DTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753709-A N-acyl-2 aryl cyclopropylmethylamine derivatives as melatonergics BRISTOL-MYERS SQUIBB COMPANY (US) 1998-05-19 US claimed
US-5889031-A CONTROLLING CIRCADIAN RHYTHMS BRISTOL-MYERS SQUIBB COMPNAY (US) 1999-03-30 US disclosed
US-5753709-A N-acyl-2 aryl cyclopropylmethylamine derivatives as melatonergics BRISTOL-MYERS SQUIBB COMPANY (US) 1998-05-19 US disclosed