SCHEMBL8335707

SCHEMBL8335707

CCOC(=O)Cc1ccc(C(=O)CCCl)cc1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.49
LMNA P02545 3/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
KMT2A Q03164 4/20 0.49
CYP4Z1 Q86W10 1/20 0.47
ALDH1A1 P00352 2/20 0.46
HPGD P15428 1/20 0.46
NPC1 O15118 2/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
RAB9A P51151 1/20 0.44
CYP4F2 P78329 1/20 0.44
CYP4A11 Q02928 1/20 0.44
KDM4E B2RXH2 1/20 0.40
TSHR P16473 1/20 0.40
HSD17B10 Q99714 1/20 0.40
POLB P06746 1/20 0.40
MEN1 O00255 1/20 0.40
HTT P42858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Methane SCHEMBL6325038 0.90 NPC1 (0.49) MAPTLMNASMN1; SMN2KMT2ACYP4Z1
SCHEMBL7335258 0.87 THRA (0.51) MAPTLMNASMN1; SMN2KMT2ACYP4Z1
SCHEMBL4268203 0.84 L3MBTL1 (0.59) MAPTLMNASMN1; SMN2KMT2ACYP4Z1
SCHEMBL15955709 0.83 KMT2A (0.60) MAPTLMNASMN1; SMN2KMT2ACYP4Z1
SCHEMBL6681547 0.82 HSD17B3 (0.58)
SCHEMBL68851 0.81 CYP4Z1 (0.62) MAPTLMNASMN1; SMN2KMT2ACYP4Z1
SCHEMBL392939 0.81 GSK3B (0.55) MAPTLMNASMN1; SMN2KMT2ACYP4Z1
SCHEMBL8149524 0.80 MAPT (0.55) MAPTLMNASMN1; SMN2KMT2ACYP4Z1
Hydrochloric Acid SCHEMBL11655187 0.79 LMNA (0.50) MAPTLMNASMN1; SMN2KMT2ACYP4Z1
SCHEMBL6393097 0.78 ALDH1A1 (0.57) MAPTLMNASMN1; SMN2KMT2ACYP4Z1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20140315881-A1 COMPOUNDS AND METHODS TEMPERO PHARMACEUTICALS, INC. 2014-10-23 US disclosed
EP-2736330-A1 COMPOUNDS AND METHODS Tempero Pharmaceuticals, Inc. (US) 2014-06-04 EP disclosed
WO-2013019682-A1 COMPOUNDS AND METHODS TEMPERO PHARMACEUTICALS, INC. (US) 2013-02-07 WO disclosed
CN-1063180-C 5H, 10H-imidazo [1, 2 -a] indeno [1, 2 -e] pyrazin-4-one derivatives, preparation thereof, and drugs containing said derivatives RHONE POULENC RORER SA (FR) 2001-03-14 CN disclosed
US-5902803-A 5H,10H-imidazo 1,2-a!indeno 1,2-e!pyrazin-4-one derivatives, preparation thereof, and drugs containing said derivatives RHONE-POULENC RORER S.A. (FR) 1999-05-11 US disclosed
CN-1180357-A 5H, 10H-imidazo [1, 2-a ] indeno [1, 2-e ] pyrazin-4-one derivatives, preparation thereof and medicaments containing same RHONE POULENC RORER SA (FR) 1998-04-29 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140315881-A1 COMPOUNDS AND METHODS RORC, RORB, RORA MAPT 3084/4885LMNA 4009/4885SMN1; SMN2 3006/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.