SCHEMBL8336244

SCHEMBL8336244

Cc1nc2cc(F)ccc2n1CCCN1CCN(c2ncc(F)cn2)CC1

nearest known ligand 0.52

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 7/20 0.52
KDM4E B2RXH2 1/20 0.49
CYP1A2 P05177 1/20 0.49
GAA P10253 1/20 0.49
CYP2C9 P11712 1/20 0.49
DRD2 P14416 1/20 0.49
HTR1A P08908 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6839501 0.85 HTR1A (0.48) HTR1A
SCHEMBL8340386 0.83 HTR7 (0.57) SIGMAR1DRD2HTR1A
SCHEMBL8788615 0.79 GRM2 (0.42) SIGMAR1DRD2HTR1A
SCHEMBL8336417 0.79 HTR3E (0.53) SIGMAR1HTR1A
SCHEMBL8341291 0.79 GRM2 (0.53) DRD2
SCHEMBL8788970 0.78 MCHR1 (0.48) SIGMAR1DRD2HTR1A
SCHEMBL9053834 0.75 DRD2 (0.50) SIGMAR1CYP1A2CYP2C9DRD2HTR1A
SCHEMBL7474002 0.75 SIGMAR1 (0.53) SIGMAR1KDM4ECYP1A2GAACYP2C9
SCHEMBL8337662 0.74 PLK1 (0.51)
SCHEMBL15748179 0.74 HTR7 (0.55) KDM4EDRD2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5889010-A PSYCHOLOGICAL DISORDERS; UROGENITAL DISORDERS; COGNITION ACTIVATORS; NERVOUS SYSTEM DISORDERS; VISION DEFECTS; CONGESTIVE HEART FAILURE; DRUG ABRUSE; PARKINSON'S DISEASE;ANTIINFLAMMATORY AGENTS; ANTIALLERGENS PFIZER INC. (US) 1999-03-30 US disclosed