SCHEMBL8337648

SCHEMBL8337648

CCOC(=O)CN(C)Cc1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.57
SMN1; SMN2 Q16637 3/20 0.57
KDM4E B2RXH2 2/20 0.57
MAPT P10636 1/20 0.57
LTA4H P09960 3/20 0.56
LMNA P02545 1/20 0.51
POLB P06746 1/20 0.51
HSD17B10 Q99714 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
NPC1 O15118 3/20 0.50
RAB9A P51151 3/20 0.50
PPID Q08752 1/20 0.48
PIN1 Q13526 1/20 0.47
ACHE P22303 1/20 0.47
TSHR P16473 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10597046 0.88 RAB9A (0.49) ALDH1A1SMN1; SMN2KDM4EMAPTLTA4H
SCHEMBL13222646 0.87 SMN1; SMN2 (0.50) ALDH1A1SMN1; SMN2KDM4EMAPTLTA4H
SCHEMBL3184733 0.86 ALDH1A1 (0.54) ALDH1A1SMN1; SMN2MAPTLTA4HLMNA
SCHEMBL29304528 0.85 LTA4H (0.55) ALDH1A1SMN1; SMN2KDM4EMAPTLTA4H
SCHEMBL254781 0.85 ALDH1A1 (0.53) ALDH1A1SMN1; SMN2MAPTLTA4HLMNA
SCHEMBL10076568 0.84 KMT2A (0.49) ALDH1A1SMN1; SMN2KDM4EMAPTLTA4H
SCHEMBL3147669 0.84 PPID (0.50) ALDH1A1SMN1; SMN2KDM4EMAPTLTA4H
SCHEMBL1303146 0.84 LTA4H (0.62) ALDH1A1SMN1; SMN2LTA4HLMNAPOLB
SCHEMBL5941081 0.83 PIN1 (0.56) ALDH1A1SMN1; SMN2LTA4HLMNAPOLB
SCHEMBL5761072 0.83 KDM4E (0.56) ALDH1A1SMN1; SMN2KDM4EMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 24 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11739072-B2 Heteroaryl compounds and their use MINORYX THERAPEUTICS S.L. (ES) 2023-08-29 US disclosed
US-11739072-B2 Heteroaryl compounds and their use MINORYX THERAPEUTICS S.L. (ES) 2023-08-29 US disclosed
US-11739072-B2 Heteroaryl compounds and their use MINORYX THERAPEUTICS S.L. (ES) 2023-08-29 US disclosed
US-20220135535-A1 HETEROARYL COMPOUNDS AND THEIR USE MINORYX THERAPEUTICS S.L. (ES) 2022-05-05 US disclosed
US-20220135535-A1 HETEROARYL COMPOUNDS AND THEIR USE MINORYX THERAPEUTICS S.L. (ES) 2022-05-05 US disclosed
EP-3562811-B1 HETEROARYL COMPOUNDS AND THEIR USE MINORYX THERAPEUTICS S L (ES) 2022-03-16 EP disclosed
US-11174242-B2 Heteroaryl compounds and their use MINORYX THERAPEUTICS S.L. (ES) 2021-11-16 US disclosed
US-11174242-B2 Heteroaryl compounds and their use MINORYX THERAPEUTICS S.L. (ES) 2021-11-16 US disclosed
WO-2020182990-A1 FUSED RING PYRIMIDONE DERIVATIVES FOR USE IN THE TREATMENT OF HBV INFECTION OR OF HBV-INDUCED DISEASES Janssen Sciences Ireland Unlimited Company (IE) 2020-09-17 WO disclosed
US-20190337922-A1 HETEROARYL COMPOUNDS AND THEIR USE MINORYX THERAPEUTICS S.L. (ES) 2019-11-07 US disclosed
US-8034949-B2 Pyrrolidine compound and a process for preparing the same MITSUBISHI TANABE PHARMA CORPORATION (JP) 2011-10-11 US disclosed
US-8034949-B2 Pyrrolidine compound and a process for preparing the same MITSUBISHI TANABE PHARMA CORPORATION (JP) 2011-10-11 US disclosed
US-20090111801-A1 SUBSTITUTED PYRAZINONE DERIVATIVES FOR USE AS A MEDICINE JANSSEN PHARMACEUTICA N.V. (BE) 2009-04-30 US disclosed
US-20090111801-A1 SUBSTITUTED PYRAZINONE DERIVATIVES FOR USE AS A MEDICINE JANSSEN PHARMACEUTICA N.V. (BE) 2009-04-30 US disclosed
WO-2007122173-A1 SUBSTITUTED PYRAZINONE DERIVATIVES FOR USE AS A MEDICINE JANSSEN PHARMACEUTICA N.V. (BE) 2007-11-01 WO disclosed
US-20070167440-A1 Novel pyrrolidine compound and a process for preparing the same MITSUBISHI TANABE PHARMA CORPORATION (JP) 2007-07-19 US disclosed
US-20070167440-A1 Novel pyrrolidine compound and a process for preparing the same MITSUBISHI TANABE PHARMA CORPORATION (JP) 2007-07-19 US disclosed
WO-2004093860-A1 INHIBITORS OF SARS RELATED CORONAVIRUS PROTEINASE PFIZER INC. (US) 2004-11-04 WO disclosed
EP-0020018-B1 CHROMAN DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM BEECHAM GROUP PLC (GB) 1983-06-01 EP disclosed
US-4303656-A ANOREXIC AGENTS BEECHAM GROUP LIMITED (GB) 1981-12-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070167440-A1 Novel pyrrolidine compound and a process for preparing the same CNR1, CNR2, OPRD1 ALDH1A1 2888/4885SMN1; SMN2 4282/4885KDM4E 535/4885
US-20090111801-A1 SUBSTITUTED PYRAZINONE DERIVATIVES FOR USE AS A MEDICINE ADRA2C, ADRB2, CHRNA5 ALDH1A1 710/4885SMN1; SMN2 432/4885KDM4E 3069/4885
US-20220135535-A1 HETEROARYL COMPOUNDS AND THEIR USE GBA1, GBA2, GAA ALDH1A1 1097/4885SMN1; SMN2 36/4885KDM4E 4446/4885
US-20190337922-A1 HETEROARYL COMPOUNDS AND THEIR USE GBA1, GBA2, GAA ALDH1A1 1097/4885SMN1; SMN2 36/4885KDM4E 4446/4885
US-11174242-B2 Heteroaryl compounds and their use GBA1, GBA2, GAA ALDH1A1 1097/4885SMN1; SMN2 36/4885KDM4E 4446/4885
US-11739072-B2 Heteroaryl compounds and their use GBA1, GBA2, GAA ALDH1A1 1097/4885SMN1; SMN2 36/4885KDM4E 4446/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.