SCHEMBL8463444

SCHEMBL8463444

COc1ccc2c(ccc(=O)n2OC(C)=O)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
ALDH1A1 P00352 2/20 0.44
HPGD P15428 2/20 0.44
HSD17B10 Q99714 1/20 0.44
PTGS2 P35354 4/20 0.43
PTGS1 P23219 3/20 0.43
AKR1C3 P42330 3/20 0.43
AKR1C2 P52895 3/20 0.43
CYP1A2 P05177 2/20 0.43
TSHR P16473 2/20 0.43
CDC42 P60953 1/20 0.43
RAC1 P63000 1/20 0.43
SLC22A6 Q4U2R8 1/20 0.43
MTNR1A P48039 1/20 0.43
MTNR1B P49286 1/20 0.43
LMNA P02545 2/20 0.42
MAPT P10636 2/20 0.42
NPC1 O15118 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27754476 0.77 MAOA (0.35) KDM4EMAPTMAOATDP1
SCHEMBL9496147 0.76 CA12 (0.50) KDM4ESMN1; SMN2L3MBTL1ALDH1A1HPGD
SCHEMBL9499012 0.76 KDM4E (0.50) KDM4ESMN1; SMN2L3MBTL1ALDH1A1HPGD
SCHEMBL28470000 0.76 TUBB1 (0.49) KDM4ESMN1; SMN2L3MBTL1ALDH1A1HPGD
SCHEMBL6074279 0.74 BRPF1 (0.59) KDM4ESMN1; SMN2L3MBTL1ALDH1A1HPGD
SCHEMBL8368861 0.72 PTGS1 (0.50) KDM4ESMN1; SMN2ALDH1A1HPGDHSD17B10
SCHEMBL4067603 0.72 KMO (0.46) KDM4ESMN1; SMN2ALDH1A1HPGDHSD17B10
SCHEMBL8366395 0.71 MAPT (0.52) KDM4ESMN1; SMN2L3MBTL1ALDH1A1HPGD
SCHEMBL4049057 0.71 GRIK1 (0.55) KDM4ESMN1; SMN2MTNR1AMTNR1BMAPT
SCHEMBL253760 0.70 GLA (0.65) KDM4ESMN1; SMN2ALDH1A1HPGDPTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850235-B1 QUINOLEIN-2(1H)-ONE DERIVATIVES AS SEROTONIN ANTAGONISTS SANOFI SYNTHELABO (FR) 1999-12-01 EP disclosed