SCHEMBL8467321

SCHEMBL8467321

CN1Cc2cc(C#CCCO)ccc2N(C(=O)OC(C)(C)C)C(CC(=O)O)C1=O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 4/20 0.35
GABRG2 P18507 4/20 0.35
GABRB3 P28472 4/20 0.35
GABRA5 P31644 4/20 0.35
GABRA3 P34903 4/20 0.35
GABRA2 P47869 4/20 0.35
GABRA6 Q16445 4/20 0.35
PRKCG P05129 1/20 0.34
PRKCB P05771 1/20 0.34
PRKCA P17252 1/20 0.34
PRKCE Q02156 1/20 0.34
PRKCD Q05655 1/20 0.34
ITGB1 P05556 1/20 0.34
ITGA4 P13612 1/20 0.34
GABRA4 P48169 3/20 0.32
GABRB2 P47870 2/20 0.32
KLK7 P49862 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
HDAC1 Q13547 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8467659 0.82 GABRG2 (0.39) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL7366878 0.81 ITGB3 (0.38) KLK7
SCHEMBL8468002 0.80 DHODH (0.37) PRKCGPRKCBPRKCAPRKCEPRKCD
SCHEMBL8323234 0.77 KLK7 (0.36) PRKCGPRKCBPRKCAPRKCEPRKCD
SCHEMBL8328325 0.70 ITGB3 (0.40) MEN1KMT2A
SCHEMBL8330616 0.69 ITGB3 (0.46)
SCHEMBL7544674 0.67 ITGB3 (0.39)
SCHEMBL5637567 0.66 DHODH (0.45) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL7798122 0.65 HSD17B3 (0.39)
SCHEMBL5637695 0.64 BRD4 (0.46) GABRA1GABRG2GABRB3GABRA5GABRA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0869787-A4 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 1999-03-24 EP disclosed
EP-0869787-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1998-10-14 EP disclosed
WO-1997024119-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-07-10 WO disclosed