SCHEMBL8330616

SCHEMBL8330616

CN1Cc2cc(CCCc3nc4ccccc4[nH]3)ccc2N(C(=O)OC(C)(C)C)C(CC(=O)O)C1=O

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 18/20 0.46
ITGAV P06756 18/20 0.46
ITGA2B P08514 3/20 0.43
CYP1A2 P05177 1/20 0.37
CYP2C9 P11712 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8323234 0.82 KLK7 (0.36) ITGB3ITGA2B
SCHEMBL8468002 0.82 DHODH (0.37) ITGB3ITGAVITGA2B
SCHEMBL8328325 0.81 ITGB3 (0.40) ITGB3ITGAVITGA2B
SCHEMBL8467842 0.77 ITGB3 (0.72) ITGB3ITGAVITGA2B
SCHEMBL8467659 0.75 GABRG2 (0.39) ITGB3ITGAVITGA2B
SCHEMBL7361297 0.75 ITGB3 (0.54) ITGB3ITGAVITGA2B
SCHEMBL7366878 0.74 ITGB3 (0.38) ITGB3ITGAVITGA2B
SCHEMBL7360585 0.70 ITGB3 (0.72) ITGB3ITGAVITGA2B
SCHEMBL8467321 0.69 GABRA1 (0.35)
SCHEMBL5486017 0.67 ITGB3 (0.65) ITGB3ITGAVITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0869787-A4 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 1999-03-24 EP disclosed
EP-0869787-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1998-10-14 EP disclosed
WO-1997024119-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-07-10 WO disclosed