SCHEMBL8323234

SCHEMBL8323234

CN1Cc2cc(CCCCC(=O)O)ccc2N(C(=O)OC(C)(C)C)C(CC(=O)O)C1=O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KLK7 P49862 7/20 0.36
KLK5 Q9Y337 6/20 0.36
PRSS1 P07477 3/20 0.36
PRSS2 P07478 3/20 0.36
PRSS3 P35030 3/20 0.36
NR1H2 P55055 4/20 0.34
RXRA P19793 3/20 0.34
NR1H3 Q13133 2/20 0.34
DHODH Q02127 1/20 0.34
PRKCA P17252 3/20 0.33
ITGB3 P05106 1/20 0.33
ITGA2B P08514 1/20 0.33
PRKCG P05129 1/20 0.33
PRKCB P05771 1/20 0.33
PRKCH P24723 1/20 0.33
PRKCE Q02156 1/20 0.33
PRKCQ Q04759 1/20 0.33
PRKCD Q05655 1/20 0.33
PLA2G10 O15496 1/20 0.33
PLA2G5 P39877 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8468002 0.93 DHODH (0.37) KLK7KLK5PRSS1PRSS2PRSS3
SCHEMBL8467659 0.84 GABRG2 (0.39) KLK7KLK5PRSS1PRSS2PRSS3
SCHEMBL7366878 0.83 ITGB3 (0.38) KLK7ITGB3ITGA2B
SCHEMBL8330616 0.82 ITGB3 (0.46) ITGB3ITGA2B
SCHEMBL8467321 0.77 GABRA1 (0.35) KLK7DHODHPRKCAPRKCGPRKCB
SCHEMBL8328325 0.71 ITGB3 (0.40) ITGB3ITGA2B
SCHEMBL7544674 0.68 ITGB3 (0.39) ITGB3ITGA2B
SCHEMBL7798122 0.66 HSD17B3 (0.39) ITGB3ITGA2B
SCHEMBL7919341 0.64 BRD4 (0.41) ITGB3ITGA2B
SCHEMBL5155939 0.64 ITGB3 (0.41) ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0869787-A4 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 1999-03-24 EP disclosed
EP-0869787-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1998-10-14 EP disclosed
WO-1997024119-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-07-10 WO disclosed