SCHEMBL8467659

SCHEMBL8467659

CN1Cc2cc(I)ccc2N(C(=O)OC(C)(C)C)C(CC(=O)O)C1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRG2 P18507 2/20 0.39
GABRB3 P28472 2/20 0.39
GABRA5 P31644 2/20 0.39
GABRA1 P14867 1/20 0.39
GABRA3 P34903 1/20 0.39
GABRA2 P47869 1/20 0.39
GABRA6 Q16445 1/20 0.39
KLK7 P49862 6/20 0.35
PLA2G10 O15496 1/20 0.34
PLA2G5 P39877 1/20 0.34
ITGB3 P05106 5/20 0.33
ITGA2B P08514 3/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
ITGAV P06756 3/20 0.33
KLK5 Q9Y337 5/20 0.32
PRSS1 P07477 2/20 0.32
PRSS2 P07478 2/20 0.32
PRSS3 P35030 2/20 0.32
ESR2 Q92731 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7366878 0.89 ITGB3 (0.38) KLK7ITGB3ITGA2BITGAV
SCHEMBL8468002 0.84 DHODH (0.37) KLK7PLA2G10PLA2G5ITGB3ITGA2B
SCHEMBL8323234 0.84 KLK7 (0.36) KLK7PLA2G10PLA2G5ITGB3ITGA2B
SCHEMBL8467321 0.82 GABRA1 (0.35) GABRG2GABRB3GABRA5GABRA1GABRA3
SCHEMBL7919362 0.82 ITGB3 (0.35) GABRG2GABRB3GABRA5GABRA1GABRA3
SCHEMBL8328325 0.76 ITGB3 (0.40) ITGB3ITGA2BMEN1KMT2AITGAV
SCHEMBL8330616 0.75 ITGB3 (0.46) ITGB3ITGA2BITGAV
SCHEMBL29294080 0.74 ACE (0.38)
SCHEMBL7544674 0.73 ITGB3 (0.39) ITGB3ITGA2BITGAV
SCHEMBL7798122 0.71 HSD17B3 (0.39) ITGB3ITGA2BITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0869787-A4 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 1999-03-24 EP disclosed
EP-0869787-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1998-10-14 EP disclosed
WO-1997024119-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-07-10 WO disclosed