SCHEMBL8517829

SCHEMBL8517829

C=CCc1ccc(C#CC(C)O)c(-c2cccnn2)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 4/20 0.36
GABRB2 P47870 4/20 0.36
MEN1 O00255 3/20 0.36
GAA P10253 3/20 0.36
MAPT P10636 3/20 0.36
KMT2A Q03164 3/20 0.36
ALDH1A1 P00352 3/20 0.36
KDM4E B2RXH2 2/20 0.36
CNR1 P21554 2/20 0.36
CNR2 P34972 2/20 0.36
ALDH2 P05091 1/20 0.36
AKR1B1 P15121 1/20 0.36
HPGD P15428 1/20 0.36
PPARG P37231 1/20 0.36
PPARD Q03181 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
TNKS O95271 1/20 0.32
PARP1 P09874 1/20 0.32
LMNA P02545 1/20 0.32
HTT P42858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8518534 0.82 LMNA (0.37) MEN1GAAMAPTKMT2AALDH1A1
SCHEMBL8517769 0.81 GABRA1 (0.39) GABRA1GABRB2MEN1GAAMAPT
SCHEMBL8517833 0.71
SCHEMBL8517770 0.68 ADRB2 (0.32) ALDH1A1KDM4ELMNA
SCHEMBL8378363 0.68 LPL (0.34)
SCHEMBL8517544 0.66 ALDH1A1 (0.41) GABRA1GABRB2MEN1GAAMAPT
SCHEMBL8601588 0.65 PTAFR (0.32)
SCHEMBL8517733 0.65 ACACB (0.40) MEN1GAAMAPTKMT2AALDH1A1
SCHEMBL8518542 0.64 ADRB2 (0.35) MAPTLMNA
SCHEMBL8516504 0.64 PTGS2 (0.41) MEN1GAAMAPTKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0628530-B1 ACETYLENE DERIVATIVES, PROCESS FOR PRODUCING THE SAME, LIQUID CRYSTAL COMPOSITION CONTAINING THE SAME AS ACTIVE INGREDIENT, AND LIQUID CRYSTAL ELEMENT MADE THEREFROM SUMITOMO CHEMICAL CO (JP) 1999-03-24 EP disclosed
US-5534188-A Acetylene derivatives, process for producing the same, liquid crystal composition containing the same as an active ingredient, and liquid crystal element using said liquid crystal composition SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1996-07-09 US disclosed
EP-0628530-A1 ACETYLENE DERIVATIVE, PROCESS FOR PRODUCING THE SAME, LIQUID CRYSTAL COMPOSITION CONTAINING THE SAME AS ACTIVE INGREDIENT, AND LIQUID CRYSTAL ELEMENT MADE THEREFROM SUMITOMO CHEMICAL COMPANY LIMITED (JP) 1994-12-14 EP disclosed