SCHEMBL8519457

SCHEMBL8519457

COc1ccc(C(=O)c2c(C)cc(CNS(=O)(=O)Cc3cccnc3)n2C)cc1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.48
SMN1; SMN2 Q16637 4/20 0.47
ALDH1A1 P00352 2/20 0.47
MMP1 P03956 1/20 0.44
MMP9 P14780 1/20 0.44
MMP13 P45452 1/20 0.44
KCNA5 P22460 1/20 0.44
ADORA2A P29274 1/20 0.43
ADORA2B P29275 1/20 0.43
NAMPT P43490 3/20 0.42
TSHR P16473 1/20 0.41
HTT P42858 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8518478 0.89 MEN1 (0.43) GAAALDH1A1NAMPTTSHRHTT
SCHEMBL8519895 0.89 ABCB11 (0.51) SMN1; SMN2ALDH1A1NAMPTTSHRHTT
Hydrochloric Acid SCHEMBL8518624 0.89 VNN1 (0.43) NAMPTTSHRHTT
SCHEMBL8519156 0.89 OPRK1 (0.46) SMN1; SMN2ALDH1A1MMP1MMP13KCNA5
Hydrochloric Acid SCHEMBL8519131 0.88 ABCB11 (0.50) SMN1; SMN2ALDH1A1NAMPTTSHRHTT
SCHEMBL8519780 0.85 LMNA (0.41) SMN1; SMN2ALDH1A1NAMPTTSHRHTT
SCHEMBL8518342 0.80 TSHR (0.43) SMN1; SMN2ALDH1A1MMP13NAMPTTSHR
SCHEMBL8518402 0.79 ABCB11 (0.47) SMN1; SMN2ALDH1A1MMP1MMP9MMP13
SCHEMBL8518393 0.78 PTGS2 (0.47) GAASMN1; SMN2ALDH1A1MMP1MMP9
SCHEMBL8519370 0.77 ABCB11 (0.46) SMN1; SMN2ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5952368-A AN INHIBITORS OF PROSTAGLANDIN G/H SYNTHASE, ANTIINFLAMMATORY AND ANALGESIC AGENTS SYNTEX (U.S.A.) INC. (US) 1999-09-14 US disclosed