Azelaic Acid

Azelaic Acid

SCHEMBL852024

O=C([O-])CCCCCCCC(=O)[O-].[Na+].[Na+]

nearest known ligand 0.65

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Azelaic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA1 known ✓ P00915 2/20 0.63
CA4 known ✓ P22748 1/20 0.47
HDAC3 O15379 3/20 0.53
HDAC1 Q13547 3/20 0.53
HDAC2 Q92769 3/20 0.53
HDAC8 Q9BY41 3/20 0.53
FFAR3 O14843 2/20 0.53
FABP3 P05413 7/20 0.52
HDAC4 P56524 1/20 0.46
HDAC7 Q8WUI4 1/20 0.46
HDAC10 Q969S8 1/20 0.46
HDAC11 Q96DB2 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
HDAC9 Q9UKV0 1/20 0.46
HDAC5 Q9UQL6 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28402678 1.00 CA1 (0.63) CA1HDAC3HDAC1HDAC2HDAC8
SCHEMBL6053545 1.00 CA1 (0.63) CA1HDAC3HDAC1HDAC2HDAC8
SCHEMBL30930281 1.00 CA1 (0.63) CA1HDAC3HDAC1HDAC2HDAC8
Pimelic Acid SCHEMBL6756717 1.00 CA1 (0.63) CA1HDAC3HDAC1HDAC2HDAC8
Sebacic Acid SCHEMBL306520 1.00 CA1 (0.63) CA1HDAC3HDAC1HDAC2HDAC8
SCHEMBL20577558 1.00 CA1 (0.63) CA1HDAC3HDAC1HDAC2HDAC8
SCHEMBL11046980 1.00 CA1 (0.63) CA1HDAC3HDAC1HDAC2HDAC8
Octanedioate SCHEMBL188028 1.00 CA1 (0.63) CA1HDAC3HDAC1HDAC2HDAC8
SCHEMBL8325989 1.00 CA1 (0.63) CA1HDAC3HDAC1HDAC2HDAC8
Sebacic Acid SCHEMBL29696252 1.00 CA1 (0.63) CA1HDAC3HDAC1HDAC2HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 197 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119488469-A Anti-drop and anti-dandruff composition and preparation method thereof 广东领秀首美生物科技有限公司 2025-02-21 CN claimed
CN-118141762-B Foam-type pharmaceutical agent and foam composition for topical application 北京罗诺强施医药技术研发中心有限公司 2024-07-12 CN claimed
CN-118141762-A Foam-type pharmaceutical agent and foam composition for topical application 北京罗诺强施医药技术研发中心有限公司 2024-06-07 CN claimed
CN-117653570-A Composition with oil control and fluffiness effects and preparation method and application thereof 珠海博御中医药研究有限公司 2024-03-08 CN claimed
CN-116585245-B Shampoo containing ginger root extract and preparation method thereof 珠海博御中医药研究有限公司 2024-02-09 CN claimed
CN-116585245-A Shampoo containing ginger root extract and preparation method thereof 珠海博御中医药研究有限公司 2023-08-15 CN claimed
CN-112080251-B Wafer grinding fluid and preparation method thereof 威科赛乐微电子股份有限公司 2022-06-10 CN claimed
CN-112795418-A Tetra-urea lubricating grease composition prepared from aromatic diamine and preparation method thereof 青岛中科润美润滑材料技术有限公司 2021-05-14 CN claimed
CN-112375607-A Tetraurea lubricating grease composition and preparation method thereof 青岛中科润美润滑材料技术有限公司 2021-02-19 CN claimed
CN-110797208-B Preparation method and application of electrode material 南京大学 2020-12-22 CN claimed
US-20160029622-A1 Plant Pathogen Resistance THE UNIVERSITY OF CHICAGO 2016-02-04 US claimed
EP-2965625-A1 PLANT PATHOGEN RESISTANCE The University of Chicago (US) 2016-01-13 EP claimed
US-9161533-B2 Plant pathogen resistance THE UNIVERSITY OF CHICAGO (US) 2015-10-20 US claimed
EP-2187736-B1 PLANT PATHOGEN RESISTANCE UNIV CHICAGO (US) 2015-07-29 EP claimed
US-20130130907-A1 PLANT PATHOGEN RESISTANCE UT-Batlelle, LLC (US) 2013-05-23 US claimed
US-8318786-B2 Plant pathogen resistance THE UNIVERSITY OF CHICAGO (US) 2012-11-27 US claimed
JP-2010536785-A 2010-12-02 JP claimed
EP-2187736-A2 PLANT PATHOGEN RESISTANCE The University of Chicago (US) 2010-05-26 EP claimed
WO-2009055126-A2 PLANT PATHOGEN RESISTANCE THE UNIVERSITY OF CHICAGO (US) 2009-04-30 WO claimed
US-20090048312-A1 PLANT PATHOGEN RESISTANCE THE UNIVERSITY OF CHICAGO (US) 2009-02-19 US claimed