SCHEMBL852151

SCHEMBL852151

[CH2][Si](C)(C)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.44
ESR2 Q92731 1/20 0.44
NR1H2 P55055 2/20 0.35
NR1H3 Q13133 2/20 0.35
TSHR P16473 4/20 0.35
LMNA P02545 1/20 0.35
ALOX12 P18054 1/20 0.35
ACHE P22303 1/20 0.35
BRD4 O60885 1/20 0.34
BRD2 P25440 1/20 0.34
MAPT P10636 2/20 0.34
PTGS1 P23219 1/20 0.33
PTGS2 P35354 1/20 0.33
NPC1 O15118 3/20 0.32
RAB9A P51151 3/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
ALDH1A1 P00352 2/20 0.32
CES2 O00748 1/20 0.31
CES1 P23141 1/20 0.31
KDM4E B2RXH2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9339604 0.81 ESR1 (0.44) ESR1ESR2NR1H2NR1H3TSHR
Water SCHEMBL28099446 0.78 ESR1 (0.67) ESR1ESR2NR1H2NR1H3TSHR
Ethylene SCHEMBL25342007 0.75 ESR1 (0.44) ESR1ESR2NR1H2NR1H3TSHR
SCHEMBL439491 0.73 ESR1 (0.36) ESR1ESR2TSHRLMNAALOX12
SCHEMBL2169977 0.73 ESR1 (0.48) ESR1ESR2NR1H2NR1H3TSHR
SCHEMBL92396 0.73 ESR1 (0.48) ESR1ESR2NR1H2NR1H3TSHR
SCHEMBL239179 0.73 ESR1 (0.48) ESR1ESR2NR1H2NR1H3TSHR
SCHEMBL63526 0.73 ESR1 (0.70) ESR1ESR2NR1H2NR1H3TSHR
SCHEMBL439492 0.73 ESR1 (0.48) ESR1ESR2NR1H2NR1H3TSHR
SCHEMBL2143198 0.73 ACHE (0.47) TSHRLMNAALOX12ACHENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 146 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1470123-A1 BICYCLIC HETEROCYCLIC SUBSTITUTED PHENYL OXAZOLIDINONE ANTIBACTERIALS, RELATED COMPOSITIONS AND METHODS Ortho-Mcneil Pharmaceutical, Inc. (US) 2004-10-27 EP claimed
US-20040067994-A1 BICYCLIC HETEROCYCLIC SUBSTITUTED PHENYL OXAZOLIDINONE ANTIBACTERIALS, AND RELATED COMPOSITIONS AND METHODS PAGET STEVEN D (US) 2004-04-08 US claimed
US-6608081-B2 Treating pneumonia ORTHO-MCNEIL PHARMACEUTICAL, INC. 2003-08-19 US claimed
WO-2003064415-A1 BICYCLIC HETEROCYCLIC SUBSTITUTED PHENYL OXAZOLIDINONE ANTIBACTERIAL, RELATED COMPOSITIONS AND METHODS ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2003-08-07 WO claimed
US-20020161029-A1 Bicyclic heterocyclic substituted phenyl oxazolidinone antibacterials, and related compositions and methods ORTHO-MCNEIL PHARMACEUTICAL, INC. 2002-10-31 US claimed
EP-0437784-B1 Imidazolidine derivatives, process for producing the same and pesticides containing the same ISHIHARA SANGYO KAISHA (JP) 1996-04-17 EP claimed
EP-0458061-B1 Agent for preserving wood and wooden materials DESOWAG MATERIALSCHUTZ GMBH (DE) 1995-10-11 EP claimed
EP-0458060-B1 Agent for preserving wood and wooden materials DESOWAG MATERIALSCHUTZ GMBH (DE) 1995-10-11 EP claimed
US-5256674-A Inecticides, miticides, nematocides ISHIHARA SANGYO KAISHA LTD. (JP) 1993-10-26 US claimed
EP-0214842-B1 ORGANOTIN COMPOUNDS AND PESTICIDES CONTAINING THEM SHIONOGI & CO., LTD. (JP) 1992-02-05 EP claimed
EP-0437784-A1 Imidazolidine derivatives, process for producing the same and pesticides containing the same ISHIHARA SANGYO KAISHA, LTD. (JP) 1991-07-24 EP claimed
US-4935408-A Organotin compounds and pesticides containing them SHIONOGI & CO., LTD. (JP) 1990-06-19 US claimed
EP-0214842-A2 Organotin compounds and pesticides containing them SHIONOGI & CO., LTD. (JP) 1987-03-18 EP claimed
JP-1170620-A None JP disclosed
EP-3604362-B1 MULTI-COMPONENT POLAR OLEFIN COPOLYMER AND METHOD FOR PRODUCING SAME JAPAN POLYETHYLENE CORP (JP) 2023-08-02 EP disclosed
US-20230132484-A1 STERICALLY HINDERED PHOSPHINE-AMIDE SUPPORTED NICKEL (II) OR PALLADIUM (II) CATALYSTS FOR THE COPOLYMERIZATION OF ETHYLENE AND POLAR COMONOMERS DOW GLOBAL TECHNOLOGIES LLC (US) 2023-05-04 US disclosed
US-4774235-A MITICIDES SHIONOGI & CO., LTD. (JP) 1988-09-27 US disclosed
EP-0214842-A2 Organotin compounds and pesticides containing them SHIONOGI & CO., LTD. (JP) 1987-03-18 EP disclosed
EP-0214842-A2 Organotin compounds and pesticides containing them SHIONOGI & CO., LTD. (JP) 1987-03-18 EP disclosed
US-4237137-A Sila-substituted 1,4-dihydropyridine derivatives and their medicinal use BAYER AKTIENGESELLSCHAFT (DE) 1980-12-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020161029-A1 Bicyclic heterocyclic substituted phenyl oxazolidinone antibacterials, and related compositions and methods OXA1L, NDUFS3, CYCS ESR1 2909/4885ESR2 1991/4885NR1H2 2006/4885
US-20040067994-A1 BICYCLIC HETEROCYCLIC SUBSTITUTED PHENYL OXAZOLIDINONE ANTIBACTERIALS, AND RELATED COMPOSITIONS AND METHODS OXA1L, NDUFS3, CYCS ESR1 2909/4885ESR2 1991/4885NR1H2 2006/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.