SCHEMBL8535748

SCHEMBL8535748

COC(=O)CCC(=O)c1ccc(C)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.63
CTNNB1 P35222 3/20 0.60
WNT3A P56704 3/20 0.60
TDP1 Q9NUW8 2/20 0.53
MEN1 O00255 3/20 0.53
NPC1 O15118 2/20 0.53
RAB9A P51151 2/20 0.53
GSK3B P49841 1/20 0.52
POLB P06746 1/20 0.51
TP53 P04637 1/20 0.51
THRB P10828 1/20 0.51
MAPT P10636 2/20 0.50
LMNA P02545 2/20 0.50
ATM Q13315 1/20 0.50
TSHR P16473 1/20 0.50
ALDH1A1 P00352 1/20 0.50
HTT P42858 1/20 0.50
HSD17B10 Q99714 1/20 0.50
PKM P14618 1/20 0.49
MMP1 P03956 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7865396 0.95 KMT2A (0.58) KMT2ACTNNB1WNT3ATDP1MEN1
SCHEMBL9077880 0.89 KMT2A (0.55) KMT2ACTNNB1WNT3ATDP1MEN1
SCHEMBL25456558 0.87 KMT2A (0.53) KMT2ACTNNB1WNT3ATDP1MEN1
SCHEMBL16552778 0.85 KMT2A (0.83) KMT2ACTNNB1WNT3AMEN1NPC1
SCHEMBL2305014 0.85 HSD17B3 (0.60) KMT2ATDP1MEN1NPC1RAB9A
SCHEMBL6388993 0.84 KMT2A (0.50) KMT2ACTNNB1WNT3ATDP1MEN1
SCHEMBL1201267 0.84 NPC1 (0.62) KMT2ACTNNB1WNT3ATDP1MEN1
SCHEMBL9263357 0.83 KMT2A (0.60) KMT2ATDP1MEN1NPC1RAB9A
SCHEMBL10749473 0.83 KMT2A (0.61) KMT2ACTNNB1WNT3ATDP1MEN1
SCHEMBL640759 0.83 LMNA (0.60) KMT2AMEN1NPC1RAB9APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 29 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119125347-A Method for detecting succinylcholine chloride intermediate and related impurities 上海旭东海普药业有限公司 2024-12-13 CN claimed
CN-119125347-A Method for detecting succinylcholine chloride intermediate and related impurities 上海旭东海普药业有限公司 2024-12-13 CN disclosed
CN-119125347-A Method for detecting succinylcholine chloride intermediate and related impurities 上海旭东海普药业有限公司 2024-12-13 CN disclosed
US-20240150343-A1 COMPOUND HAVING BRD4 INHIBITORY ACTIVITY, PREPARATION METHOD THEREFOR AND USE THEREOF HAIHE BIOPHARMA CO., LTD. (CN) 2024-05-09 US disclosed
EP-4043462-A1 COMPOUND HAVING BRD4 INHIBITORY ACTIVITY, PREPARATION METHOD THEREFOR AND USE THEREOF Haihe Biopharma Co., Ltd. (CN) 2022-08-17 EP disclosed
CN-114401964-A Compound with BRD4 inhibitory activity, preparation method and application thereof 上海海和药物研究开发股份有限公司 2022-04-26 CN disclosed
WO-2021068755-A1 COMPOUND HAVING BRD4 INHIBITORY ACTIVITY, PREPARATION METHOD THEREFOR AND USE THEREOF 上海海和药物研究开发股份有限公司 2021-04-15 WO disclosed
WO-2021068755-A1 COMPOUND HAVING BRD4 INHIBITORY ACTIVITY, PREPARATION METHOD THEREFOR AND USE THEREOF 上海海和药物研究开发股份有限公司 2021-04-15 WO disclosed
CN-112625036-A Compound with BRD4 inhibitory activity, preparation method and application thereof 上海海和药物研究开发股份有限公司 2021-04-09 CN disclosed
US-8367662-B2 Organic compounds NOVARTIS AG (CH) 2013-02-05 US disclosed
US-20090197795-A1 PREPARATION AND USE OF ARYL ALKYL ACID DERIVATIVES FOR THE TREATMENT OF OBESITY BAYER HEALTHCARE LLC (US) 2009-08-06 US disclosed
US-20090176777-A1 Imidazo (1,2-a)Pyridin-3-YL-Acetic Acid Hydrazides, Proesses for Their Preparation and Pharmaceutical Uses Thereof FERRER INTERNACIONAL, S.A. (ES) 2009-07-09 US disclosed
US-20090176777-A1 Imidazo (1,2-a)Pyridin-3-YL-Acetic Acid Hydrazides, Proesses for Their Preparation and Pharmaceutical Uses Thereof FERRER INTERNACIONAL, S.A. (ES) 2009-07-09 US disclosed
EP-1973907-B1 IMIDAZO (1,2-A)PYRIDIN-3-YL-ACETIC ACID HYDRAZIDES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL USES THEREOF FERRER INT (ES) 2009-05-06 EP disclosed
US-7423156-B2 Preparation and use of aryl alkyl acid derivatives for the treatment of obesity BAYER PHARMACEUTICALS CORPORATION (US) 2008-09-09 US disclosed
WO-2007077159-A1 IMIDAZO (1,2-A)PYRIDIN-3-YL-ACETIC ACID HYDRAZIDES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL USES THEREOF FERRER INTERNACIONAL, S.A. (ES) 2007-07-12 WO disclosed
EP-1803722-A1 Imidazo[1,2-a]pyridin-3-yl-acetic acid hydrazides, processes for their preparation and pharmaceutical uses thereof FERRER INTERNACIONAL, S.A. (ES) 2007-07-04 EP disclosed
EP-0885869-A1 THERAPEUTIC AGENT FOR DIABETES Japan Tobacco Inc. (JP) 1998-12-23 EP disclosed
WO-1992018484-A1 3-AMINO-5-ARYLPYRAZOLE-4-ACETIC ACID DERIVATIVES EXHIBITING THERAPEUTIC EFFECTS A.H. ROBINS COMPANY, INCORPORATED (US) 1992-10-29 WO disclosed
US-5057534-A Anxiolytic, anticonfulsant and muscle relaxants A. H. ROBINS COMPANY INCORPORATED (US) 1991-10-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240150343-A1 COMPOUND HAVING BRD4 INHIBITORY ACTIVITY, PREPARATION METHOD THEREFOR AND USE THEREOF BRD4, BICRA, BET1 KMT2A 326/4885CTNNB1 1845/4885WNT3A 1586/4885
US-20090197795-A1 PREPARATION AND USE OF ARYL ALKYL ACID DERIVATIVES FOR THE TREATMENT OF OBESITY FABP4, GPR119, LIPC KMT2A 627/4885CTNNB1 2704/4885WNT3A 1596/4885
US-20090176777-A1 Imidazo (1,2-a)Pyridin-3-YL-Acetic Acid Hydrazides, Proesses for Their Preparation and Pharmaceutical Uses Thereof GABRA3, GABRA1, GABRA2 KMT2A 895/4885CTNNB1 3563/4885WNT3A 2556/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.