SCHEMBL8539384

SCHEMBL8539384

COc1ccccc1C1CNc2ccccc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 3/20 0.47
ALDH1A1 P00352 2/20 0.46
HPGD P15428 2/20 0.46
TDP1 Q9NUW8 2/20 0.46
KDM4E B2RXH2 1/20 0.46
GAA P10253 1/20 0.46
MAPT P10636 1/20 0.46
HTT P42858 1/20 0.46
MEN1 O00255 1/20 0.42
USP2 O75604 1/20 0.42
KMT2A Q03164 1/20 0.42
CYP19A1 P11511 1/20 0.42
LMNA P02545 1/20 0.42
TSHR P16473 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
PKM P14618 1/20 0.42
HTR2A P28223 1/20 0.41
HTR2B P41595 1/20 0.41
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8482343 0.85 PKM (0.43) HTR2CALDH1A1HPGDTDP1KDM4E
SCHEMBL12960809 0.78 HTR1A (0.46) HTR2CALDH1A1MEN1USP2KMT2A
SCHEMBL8540456 0.77 PAX8 (0.47) ALDH1A1KDM4EGAAMAPTMEN1
SCHEMBL8130957 0.73 GID4 (0.53) HTR2CKDM4EGAAMEN1KMT2A
SCHEMBL8493961 0.73 MEN1 (0.42) HTR2CALDH1A1HPGDTDP1KDM4E
SCHEMBL4001774 0.72 MEN1 (0.52) ALDH1A1HPGDTDP1KDM4EMAPT
Hydrochloric Acid SCHEMBL11553849 0.71 MEN1 (0.50) HPGDKDM4EGAAMAPTMEN1
SCHEMBL25044117 0.71 HTR2C (0.68) HTR2CMEN1USP2KMT2AL3MBTL1
SCHEMBL5871368 0.70 PRCP (0.42) HTR2CGAAMAPTMEN1KMT2A
SCHEMBL10690101 0.69 ALDH1A1 (0.48) ALDH1A1HPGDTDP1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1204121-C 1,4-substituted cyclic amine derivatives EISAI CO LTD (JP) 2005-06-01 CN disclosed
CN-1253547-A 1,4-substituted cyclic amine derivatives EISAI CO LTD (JP) 2000-05-17 CN disclosed
EP-0721949-B1 INDOLINE COMPOUND AND 5-HT 3? RECEPTOR ANTAGONIST CONTAINING THE SAME AS ACTIVE INGREDIENT TOKYO TANABE CO (JP) 1998-01-07 EP disclosed
US-5677326-A GASTROINTESTINAL DISORDERS TOKYO TANABE COMPANY LIMITED (JP) 1997-10-14 US disclosed
EP-0721949-A1 INDOLINE COMPOUND AND 5-HT 3? RECEPTOR ANTAGONIST CONTAINING THE SAME AS ACTIVE INGREDIENT TOKYO TANABE COMPANY LIMITED (JP) 1996-07-17 EP disclosed