SCHEMBL8540305

SCHEMBL8540305

COc1ccc(CCC(=O)N2CCC(CCn3ccnc3)CC2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FKBP1A P62942 1/20 0.52
KMT2A Q03164 5/20 0.52
ALDH1A1 P00352 5/20 0.52
TSHR P16473 3/20 0.52
MEN1 O00255 3/20 0.47
CYP19A1 P11511 1/20 0.47
KDM4E B2RXH2 1/20 0.47
ME2 P23368 1/20 0.46
ME1 P48163 1/20 0.46
ME3 Q16798 1/20 0.46
LMNA P02545 2/20 0.44
GAA P10253 1/20 0.44
PKM P14618 1/20 0.44
HTT P42858 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
C3AR1 Q16581 1/20 0.44
TP53 P04637 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8545661 0.89 GRIN2B (0.46) KMT2AALDH1A1MEN1CYP19A1C3AR1
SCHEMBL8540403 0.87 TBXAS1 (0.46) KMT2AMEN1CYP19A1ME2ME1
SCHEMBL8540312 0.86 GRIN2B (0.55) FKBP1AALDH1A1TSHRKDM4ECPB1
SCHEMBL8540293 0.86 CPB1 (0.44) CYP2D6CPB1
SCHEMBL8703355 0.82 PKM (0.55) FKBP1AKMT2AALDH1A1TSHRMEN1
SCHEMBL8543266 0.81 CYP3A4 (0.52) KMT2AALDH1A1TSHRMEN1LMNA
SCHEMBL8538696 0.81 FAAH (0.50) ALDH1A1MEN1KDM4ECPB1
SCHEMBL8541116 0.81 FAAH (0.57) ALDH1A1KDM4ESMN1; SMN2CPB1TDP1
SCHEMBL9031024 0.78 PKM (0.53) KMT2AALDH1A1MEN1KDM4ELMNA
SCHEMBL9030298 0.77 C5AR1 (0.48) KMT2ATSHRMEN1LMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0705258-B1 AZOLYL-CYCLIC AMINE DERIVATIVES WITH IMMUNOMODULATORY ACTIVITY KNOLL AG (DE) 1998-12-30 EP disclosed
EP-0705258-A1 AZOLYL-CYCLIC AMINE DERIVATIVES WITH IMMUNOMODULATORY ACTIVITY Knoll AG (DE) 1996-04-10 EP disclosed
WO-1995000507-A1 AZOLYL-CYCLIC AMINE DERIVATIVES WITH IMMUNOMODULATORY ACTIVITY KNOLL AG (DE) 1995-01-05 WO disclosed