SCHEMBL8540403

SCHEMBL8540403

O=C(CCc1ccc(Cl)cc1)N1CCC(CCn2ccnc2)CC1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 2/20 0.46
CPB1 P15086 1/20 0.45
FAAH O00519 2/20 0.44
CYP2A6 P11509 1/20 0.44
CYP19A1 P11511 1/20 0.44
CYP11B1 P15538 1/20 0.44
CYP11B2 P19099 1/20 0.44
CYP2B6 P20813 1/20 0.44
ME2 P23368 1/20 0.43
ME1 P48163 1/20 0.43
ME3 Q16798 1/20 0.43
GRIN2B Q13224 1/20 0.43
C3AR1 Q16581 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
MEN1 O00255 1/20 0.43
MAPT P10636 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8545661 0.89 GRIN2B (0.46) TBXAS1CPB1FAAHCYP19A1CYP11B1
SCHEMBL8540312 0.89 GRIN2B (0.55) TBXAS1CPB1FAAHGRIN2B
SCHEMBL8540305 0.87 FKBP1A (0.52) CPB1CYP19A1ME2ME1ME3
SCHEMBL8540293 0.87 CPB1 (0.44) TBXAS1CPB1FAAHGRIN2BCYP2D6
SCHEMBL9031263 0.83 F10 (0.52) CPB1FAAHGRIN2BC3AR1MEN1
SCHEMBL8541116 0.83 FAAH (0.57) TBXAS1CPB1FAAHGRIN2B
SCHEMBL8538696 0.83 FAAH (0.50) TBXAS1CPB1FAAHGRIN2BMEN1
SCHEMBL8695119 0.82 L3MBTL1 (0.53) CYP2A6CYP19A1CYP11B1CYP11B2CYP2B6
SCHEMBL8544284 0.80 CYP19A1 (0.49) TBXAS1CYP2A6CYP19A1CYP11B1CYP11B2
SCHEMBL9031024 0.80 PKM (0.53) CPB1FAAHGRIN2BC3AR1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0705258-B1 AZOLYL-CYCLIC AMINE DERIVATIVES WITH IMMUNOMODULATORY ACTIVITY KNOLL AG (DE) 1998-12-30 EP disclosed
US-5741800-A ANTIINFLAMMATORY AGENT, ANTIALLERGENS KNOLL AKTIENGESELLACHAFT (DE) 1998-04-21 US disclosed
WO-1995000507-A1 AZOLYL-CYCLIC AMINE DERIVATIVES WITH IMMUNOMODULATORY ACTIVITY KNOLL AG (DE) 1995-01-05 WO disclosed