SCHEMBL8546281

SCHEMBL8546281

COc1ccc2c(CCC(=O)O)c(C(=O)c3ccc(C#N)cc3)oc2c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.58
SMN1; SMN2 Q16637 3/20 0.58
CYP3A4 P08684 2/20 0.58
CNR1 P21554 2/20 0.58
CNR2 P34972 2/20 0.58
ALOX15 P16050 1/20 0.58
CASP1 P29466 1/20 0.58
CASP7 P55210 1/20 0.58
KDM4E B2RXH2 7/20 0.45
ALDH1A1 P00352 5/20 0.45
HSD17B10 Q99714 3/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
MEN1 O00255 1/20 0.44
LMNA P02545 1/20 0.44
KMT2A Q03164 1/20 0.44
TUBB4A P04350 1/20 0.43
TUBB P07437 1/20 0.43
TUBA3C P0DPH7 1/20 0.43
TUBA1B P68363 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8549320 0.78 MAPT (0.46) MAPTSMN1; SMN2CYP3A4CNR1CNR2
SCHEMBL8324883 0.75 NPC1 (0.48) MAPTSMN1; SMN2CYP3A4KDM4EALDH1A1
SCHEMBL5225465 0.74 SLC22A12 (0.52) MAPTSMN1; SMN2CYP3A4CNR1CNR2
SCHEMBL3736014 0.73 CNR2 (1.00) MAPTSMN1; SMN2CYP3A4CNR1CNR2
SCHEMBL8544863 0.73 KDM4E (0.58) MAPTSMN1; SMN2CASP1CASP7KDM4E
SCHEMBL8550683 0.71 DGAT2 (0.41) MAPTSMN1; SMN2CYP3A4KDM4EALDH1A1
SCHEMBL7123280 0.71 CNR2 (0.90) MAPTSMN1; SMN2CYP3A4CNR1CNR2
SCHEMBL8543822 0.70 CASP1 (0.52) MAPTSMN1; SMN2CASP1CASP7KDM4E
SCHEMBL4437800 0.70 ALDH1A1 (0.52) MAPTSMN1; SMN2CASP1CASP7KDM4E
SCHEMBL16541126 0.70 MAPT (0.61) MAPTSMN1; SMN2KDM4EALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5504213-A ANTIINFLAMMATORY AGENTS BAYER AKTIENGESELLSCHAFT (DE) 1996-04-02 US claimed
EP-0623607-B1 Benzofuranyl-and-thiophenyl-alkanecarboxyclic acid derivatives BAYER AG (DE) 1998-07-15 EP disclosed
US-5504213-A ANTIINFLAMMATORY AGENTS BAYER AKTIENGESELLSCHAFT (DE) 1996-04-02 US disclosed
EP-0623607-A1 Benzofuranyl-and-thiophenyl-alkanecarboxyclic acid derivatives BAYER AG (DE) 1994-11-09 EP disclosed