SCHEMBL8549068

SCHEMBL8549068

CC(=O)c1ccc(N2CCN(C(C)CN(O)C(=O)c3ccc4c(c3)CCOC4)CC2)cc1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.39
TDP1 Q9NUW8 1/20 0.39
ALDH1A1 P00352 7/20 0.38
MAPT P10636 8/20 0.38
TSHR P16473 1/20 0.38
ATM Q13315 1/20 0.37
SMN1; SMN2 Q16637 3/20 0.36
KDM4E B2RXH2 3/20 0.36
KMT2A Q03164 4/20 0.35
HIF1A Q16665 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
RAD52 P43351 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8552472 0.89 MAPT (0.40) ALDH1A1MAPTSMN1; SMN2RAD52
SCHEMBL8550687 0.77 DRD4 (0.48) POLBTDP1ALDH1A1MAPTTSHR
SCHEMBL8551580 0.76 ALDH1A1 (0.38) ALDH1A1MAPTSMN1; SMN2KMT2ANPC1
SCHEMBL8549102 0.73 SMN1; SMN2 (0.39) ALDH1A1MAPTSMN1; SMN2KMT2ANPC1
SCHEMBL8550140 0.73 NAMPT (0.45) ALDH1A1MAPTSMN1; SMN2
SCHEMBL8549327 0.70 DRD2 (0.39) POLBTDP1ALDH1A1MAPTSMN1; SMN2
SCHEMBL8549471 0.70 DRD4 (0.48) MAPT
SCHEMBL8551575 0.70 DRD4 (0.48) ALDH1A1
SCHEMBL8553551 0.70 DRD4 (0.48)
SCHEMBL8550252 0.69 DRD4 (0.59) POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0836599-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1998-04-22 EP claimed
EP-0836599-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1998-04-22 EP disclosed