SCHEMBL8551580

SCHEMBL8551580

CC(CNC(=O)c1ccc2c(c1)CCOC2)N1CCN(c2ccc(C(=O)N(C)C)cc2)CC1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
PRMT5 O14744 3/20 0.38
TP53 P04637 2/20 0.38
OPRM1 P35372 1/20 0.38
OPRD1 P41143 1/20 0.38
MAPT P10636 5/20 0.37
LMNA P02545 3/20 0.37
NPC1 O15118 1/20 0.37
HDAC3 O15379 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
KMT2A Q03164 3/20 0.37
MEN1 O00255 2/20 0.37
PKM P14618 1/20 0.37
WDR77 Q9BQA1 2/20 0.36
HTR1D P28221 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8549102 0.88 SMN1; SMN2 (0.39) ALDH1A1SMN1; SMN2PRMT5TP53MAPT
SCHEMBL8550140 0.88 NAMPT (0.45) ALDH1A1SMN1; SMN2PRMT5TP53MAPT
SCHEMBL8549479 0.84 HTR1A (0.50) MAPT
SCHEMBL8627748 0.83 MEN1 (0.45) ALDH1A1SMN1; SMN2TP53MAPTLMNA
SCHEMBL8553947 0.80 AKR1C3 (0.41) ALDH1A1SMN1; SMN2TP53MAPTLMNA
SCHEMBL8549068 0.76 POLB (0.39) ALDH1A1SMN1; SMN2MAPTNPC1KMT2A
SCHEMBL8549848 0.76 DRD2 (0.43) PRMT5TP53OPRM1MAPTLMNA
SCHEMBL8551575 0.76 DRD4 (0.48) ALDH1A1HTR1D
SCHEMBL8552472 0.74 MAPT (0.40) ALDH1A1SMN1; SMN2MAPTLMNA
SCHEMBL7092149 0.73 DRD2 (0.40) ALDH1A1SMN1; SMN2MAPTLMNANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0836599-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1998-04-22 EP disclosed