SCHEMBL8549102

SCHEMBL8549102

CCC(=O)c1ccc(N2CCN(C(C)CNC(=O)c3ccc4c(c3)CCOC4)CC2)cc1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.39
ALDH1A1 P00352 2/20 0.39
PRMT5 O14744 1/20 0.39
TP53 P04637 2/20 0.38
RAD52 P43351 1/20 0.38
MAPT P10636 7/20 0.37
LMNA P02545 3/20 0.37
NPC1 O15118 1/20 0.37
HDAC3 O15379 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
KMT2A Q03164 3/20 0.37
MEN1 O00255 2/20 0.37
PKM P14618 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
HTR1D P28221 1/20 0.36
ABCB1 P08183 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8550140 0.90 NAMPT (0.45) SMN1; SMN2ALDH1A1PRMT5TP53MAPT
SCHEMBL8551580 0.88 ALDH1A1 (0.38) SMN1; SMN2ALDH1A1PRMT5TP53MAPT
SCHEMBL8627748 0.84 MEN1 (0.45) SMN1; SMN2ALDH1A1TP53MAPTLMNA
SCHEMBL8550457 0.83 HTR1A (0.51) MAPT
SCHEMBL8553947 0.81 AKR1C3 (0.41) SMN1; SMN2ALDH1A1TP53MAPTLMNA
SCHEMBL8549848 0.77 DRD2 (0.43) PRMT5TP53MAPTLMNA
SCHEMBL8549100 0.73 DRD4 (0.47) SMN1; SMN2MAPTKMT2AMEN1HTR1D
SCHEMBL8549068 0.73 POLB (0.39) SMN1; SMN2ALDH1A1RAD52MAPTNPC1
SCHEMBL8548777 0.73 HTR1D (0.54) HTR1D
SCHEMBL8553219 0.72 HTR1A (0.52) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0836599-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1998-04-22 EP claimed
EP-0836599-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1998-04-22 EP disclosed