SCHEMBL8552472

SCHEMBL8552472

CC(CN(O)C(=O)c1ccc2c(c1)CCOC2)N1CCN(c2ccc(C(F)(F)F)cc2)CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.40
LMNA P02545 1/20 0.40
HTR1A P08908 2/20 0.40
AKR1C3 P42330 1/20 0.40
RORC P51449 1/20 0.35
SLC6A9 P48067 1/20 0.35
CA12 O43570 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35
RAD52 P43351 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
MMP2 P08253 2/20 0.34
MMP9 P14780 2/20 0.34
MMP3 P08254 1/20 0.34
MMP8 P22894 1/20 0.34
MMP13 P45452 1/20 0.34
ALDH1A1 P00352 1/20 0.34
GAA P10253 1/20 0.34
SLC2A1 P11166 1/20 0.34
LRRK2 Q5S007 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8549068 0.89 POLB (0.39) MAPTRAD52SMN1; SMN2ALDH1A1
SCHEMBL8549843 0.79 DRD4 (0.46) MAPTLMNAHTR1AAKR1C3RORC
SCHEMBL8551580 0.74 ALDH1A1 (0.38) MAPTLMNASMN1; SMN2ALDH1A1
SCHEMBL8554330 0.73 CD274 (0.59) HTR1A
SCHEMBL8550140 0.72 NAMPT (0.45) MAPTLMNASMN1; SMN2ALDH1A1
SCHEMBL8549102 0.71 SMN1; SMN2 (0.39) MAPTLMNARAD52SMN1; SMN2ALDH1A1
SCHEMBL8550849 0.70 DRD4 (0.46) MAPTLMNAHTR1A
SCHEMBL8549507 0.70 HTR7 (0.45) MAPTGAA
SCHEMBL8549327 0.69 DRD2 (0.39) MAPTLMNAHTR1AAKR1C3SMN1; SMN2
SCHEMBL8550263 0.68 DRD4 (0.48) HTR1ARORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0836599-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1998-04-22 EP claimed