SCHEMBL8549558

SCHEMBL8549558

N#CCc1c[nH]c2ccc(OCc3ccccc3)c(Cl)c12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.45
IMPDH2 P12268 1/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
ATP4A P20648 1/20 0.39
MAPK1 P28482 1/20 0.39
ATP4B P51164 1/20 0.39
BLM P54132 1/20 0.39
PMP22 Q01453 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
TRPM8 Q7Z2W7 3/20 0.39
KDM4E B2RXH2 1/20 0.39
MAPT P10636 1/20 0.39
LTA4H P09960 3/20 0.38
PLA2G2A P14555 3/20 0.38
HTR1D P28221 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5265155 0.84 HTR2A (0.62) HTR2AIMPDH2MEN1KMT2ACYP1A2
SCHEMBL8869470 0.82 CSNK2A1 (0.38) HTR2AMEN1KMT2ACYP1A2CYP3A4
SCHEMBL8543015 0.81 TRPM8 (0.56) HTR2ACYP1A2CYP3A4CYP2D6TRPM8
Hydrochloric Acid SCHEMBL8547802 0.81 LTA4H (0.57) HTR2APMP22TRPM8KDM4EMAPT
SCHEMBL8545281 0.81 HTR2A (0.56) HTR2AMEN1KMT2ACYP3A4CYP2D6
SCHEMBL8544872 0.80 CSNK2A1 (0.38) HTR2ACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8548477 0.79 HTR1A (0.42) HTR2ACSNK2A1HTR6
SCHEMBL8549571 0.79 HTR1B (0.37) HTR2AMEN1KMT2ACYP1A2CYP3A4
SCHEMBL8544006 0.79 HTR2A (0.73) HTR2ATRPM8HTR1DSLC6A4HTR6
Hydrochloric Acid SCHEMBL8549336 0.78 HTR2A (0.71) HTR2ATRPM8LTA4HPLA2G2AHTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0593513-B1 TRYPTAMINE ANALOGUES, THEIR SYNTHESIS AND THEIR USE AS 5-HT1-LIKE RECEPTORS OR 5-HT2 RECEPTOR AGONISTES SMITHKLINE BEECHAM PLC (GB) 1998-10-28 EP disclosed
US-5571833-A TREATMENT OF MIGRAINE, PORTAL HYPERTENSION SMITHKLINE BEECHAM PLC (GB) 1996-11-05 US disclosed
EP-0593513-A1 TRYPTAMINE ANALOGUES, THEIR SYNTHESIS AND THEIR USE AS 5-HT1-LIKE RECEPTORS OR 5-HT2 RECEPTOR AGONISTES SMITHKLINE BEECHAM PLC (GB) 1994-04-27 EP disclosed
WO-1993000333-A1 TRYPTAMINE ANALOGUES, THEIR SYNTHESIS AND THEIR USE AS 5-HT1-LIKE OR 5-HT2 RECEPTOR AGONISTS SMITHKLINE BEECHAM PLC (GB) 1993-01-07 WO disclosed