SCHEMBL8553335

SCHEMBL8553335

CN(CCO)c1nc(Nc2ccccc2)nc(C(=C(N)c2ccccc2S(=O)(=O)[O-])c2ccccc2S(=O)(=O)[O-])n1.[Na+].[Na+]

nearest known ligand 0.53

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CA1 known ✓ P00915 10/20 0.53
CA2 known ✓ P00918 10/20 0.53
CA12 known ✓ O43570 6/20 0.53
CA9 Q16790 10/20 0.53
ALDH1A1 P00352 1/20 0.36
NPSR1 Q6W5P4 1/20 0.33
RECQL P46063 1/20 0.33
MCL1 Q07820 1/20 0.33
MAPT P10636 1/20 0.32
CDK5 Q00535 1/20 0.32
CDK5R1 Q15078 1/20 0.32
EGFR P00533 1/20 0.32
KCNH3 Q9ULD8 1/20 0.31
TAAR1 Q96RJ0 1/20 0.31
NPY5R Q15761 1/20 0.31
SLC2A1 P11166 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7098829 0.85 CA1 (0.57) CA1CA2CA9CA12ALDH1A1
SCHEMBL8534511 0.79 RECQL (0.36) CA1CA2CA9CA12NPSR1
SCHEMBL8318080 0.78 CA1 (0.48) CA1CA2CA9CA12ALDH1A1
SCHEMBL30396962 0.77 CA1 (0.55) CA1CA2CA9CA12ALDH1A1
SCHEMBL30880453 0.75 CA1 (0.44) CA1CA2CA9CA12ALDH1A1
SCHEMBL8582932 0.75 CA1 (0.44) CA1CA2CA9CA12ALDH1A1
SCHEMBL3144480 0.74 CA1 (0.55) CA1CA2CA9CA12ALDH1A1
SCHEMBL344719 0.74 CA1 (0.55) CA1CA2CA9CA12ALDH1A1
SCHEMBL29404788 0.74 CA1 (0.55) CA1CA2CA9CA12ALDH1A1
SCHEMBL29351875 0.74 CA1 (0.55) CA1CA2CA9CA12ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5861370-A DIESTER QUATERNARY AMMONIUM COMPOUND, PERFUME, LOW MOLECULAR WEIGHT ALCOHOL, ORGANINC SOLVENT AND DISPERSING AID THE PROCTER & GAMBLE COMPANY (US) 1999-01-19 US disclosed