SCHEMBL8554087

SCHEMBL8554087

CCC(O)CC(c1ccc(-c2cccc(C(C)=O)c2)cc1)c1cccnc1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 2/20 0.46
KCNH2 Q12809 1/20 0.46
SUCNR1 Q9BXA5 2/20 0.46
ADRB1 P08588 2/20 0.44
ADRB3 P13945 2/20 0.44
ADRB2 P07550 1/20 0.44
KMO O15229 1/20 0.44
FFAR1 O14842 1/20 0.44
CYP17A1 P05093 1/20 0.42
PDE4D Q08499 1/20 0.42
FYN P06241 1/20 0.41
ALDH1A1 P00352 1/20 0.40
HTT P42858 1/20 0.40
AKR1C3 P42330 2/20 0.40
AKR1C2 P52895 2/20 0.40
CTSA P10619 1/20 0.39
LMNA P02545 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8550753 0.81 TBXAS1 (0.45) ADRB1ADRB3PDE4DALDH1A1HTT
SCHEMBL8551240 0.75 SMN1; SMN2 (0.44) KCNA5ADRB1ADRB3ADRB2CYP17A1
SCHEMBL8555638 0.75 SUCNR1 (0.43) KCNA5KCNH2SUCNR1ADRB1ADRB3
SCHEMBL8478810 0.75 MMP12 (0.48) ADRB1ADRB3ADRB2KMOFYN
SCHEMBL4426460 0.73 KMO (0.73) KMOFYNALDH1A1HTT
SCHEMBL8555195 0.72 KCNA5 (0.45) KCNA5SUCNR1FFAR1CYP17A1PDE4D
Hydrochloric Acid SCHEMBL8555644 0.70 CYP3A4 (0.44) KCNH2CYP17A1PDE4DLMNASMN1; SMN2
SCHEMBL8552254 0.70 SUCNR1 (0.50) KCNA5SUCNR1FFAR1CYP17A1PDE4D
SCHEMBL8551012 0.69 PDE4D (0.47) KCNA5KCNH2CYP17A1PDE4DAKR1C3
SCHEMBL8551743 0.69 KMO (0.51) KCNA5KCNH2SUCNR1ADRB1ADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0865431-A2 COMPOUNDS Astra Pharmaceuticals Limited (GB) 1998-09-23 EP disclosed
WO-1997020815-A1 COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1997-06-12 WO disclosed