SCHEMBL8554263

SCHEMBL8554263

CCCc1[nH]c2cc(C(N)=O)cc(Cc3ccccc3Cl)c2c1C(=O)N(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 2/20 0.39
LMNA P02545 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
ALDH1A1 P00352 1/20 0.36
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
SIRT1 Q96EB6 1/20 0.35
PTGES O14684 1/20 0.35
CNR1 P21554 1/20 0.35
POLB P06746 1/20 0.34
RORC P51449 1/20 0.34
HAT1 O14929 1/20 0.34
EP300 Q09472 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
ATM Q13315 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
MAPT P10636 1/20 0.34
P2RX7 Q99572 1/20 0.34
SLC6A2 P23975 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6930961 0.88 ALOX5 (0.39) ALOX5LMNASMN1; SMN2ALDH1A1PDE3B
SCHEMBL8551861 0.88 ALOX5 (0.41) ALOX5LMNASMN1; SMN2ALDH1A1PDE3B
SCHEMBL251645 0.81 ALOX5 (0.43) ALOX5LMNASMN1; SMN2ALDH1A1PDE3B
SCHEMBL8551585 0.79 SMN1; SMN2 (0.48) ALOX5LMNASMN1; SMN2ALDH1A1PDE3B
SCHEMBL8555588 0.78 SMN1; SMN2 (0.47) ALOX5LMNASMN1; SMN2ALDH1A1PDE3B
SCHEMBL7424550 0.77 ALOX5 (0.39) ALOX5LMNASMN1; SMN2ALDH1A1PDE3B
SCHEMBL8554409 0.77 LMNA (0.47) ALOX5LMNASMN1; SMN2PDE3BPDE3A
SCHEMBL8558633 0.76 ALOX5 (0.40) ALOX5LMNASMN1; SMN2ALDH1A1PDE3B
Hydrochloric Acid SCHEMBL8627726 0.75 ALOX5 (0.40) ALOX5LMNASMN1; SMN2ALDH1A1PDE3B
SCHEMBL7707708 0.74 KMT2A (0.41) LMNASMN1; SMN2ALDH1A1PDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0820441-A1 INDOLE DERIVATIVES AS cGMP-PDE INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-01-28 EP disclosed