SCHEMBL8562455

SCHEMBL8562455

CCOc1cc2c(O)cc(C)nc2nc1C

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 4/20 0.34
ALDH1A1 P00352 5/20 0.34
KDM4E B2RXH2 3/20 0.34
HPGD P15428 3/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
CYP1A2 P05177 1/20 0.34
TSHR P16473 1/20 0.34
HSD17B10 Q99714 1/20 0.34
ADORA1 P30542 2/20 0.33
ALOX5 P09917 1/20 0.33
MAPK1 P28482 1/20 0.33
ADORA2A P29274 1/20 0.33
MEN1 O00255 5/20 0.33
KMT2A Q03164 5/20 0.33
TP53 P04637 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
ESR1 P03372 1/20 0.33
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32
PKM P14618 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8567944 0.81 KDM4E (0.38) GAAALDH1A1KDM4EHPGDSMN1; SMN2
SCHEMBL8329040 0.80 KMT2A (0.39) GAAALDH1A1KDM4EHPGDSMN1; SMN2
SCHEMBL8565727 0.75 KDM4E (0.33) GAAALDH1A1KDM4EHPGDSMN1; SMN2
SCHEMBL8561182 0.73 HSD17B10 (0.36) GAAALDH1A1KDM4EHPGDSMN1; SMN2
SCHEMBL8565860 0.70 POLB (0.54) ALDH1A1SMN1; SMN2CYP1A2MAPK1MEN1
SCHEMBL8324245 0.70 TSHR (0.42) ALDH1A1KDM4EHPGDSMN1; SMN2CYP1A2
Hydrochloric Acid SCHEMBL8567040 0.69 LMNA (0.54) ALDH1A1SMN1; SMN2CYP1A2TSHRHSD17B10
SCHEMBL8322260 0.69 DPP4 (0.48) KDM4ETSHRMAPT
SCHEMBL8328855 0.69 DPP4 (0.40) TSHRMAPK1LMNA
SCHEMBL8562829 0.68 ALDH1A1 (0.38) ALDH1A1HPGDTSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0618916-B1 ANTI-RHEUMATIC NAPHTHYRIDINE DERIVATIVES KNOLL AG (DE) 1998-09-23 EP disclosed
US-5464781-A TREATING RHEUMATIC DISEASES THE BOOTS COMPANY PLC (GB) 1995-11-07 US disclosed
EP-0618916-A1 ANTI-RHEUMATIC NAPHTHYRIDINE DERIVATIVES Knoll AG (DE) 1994-10-12 EP disclosed
WO-1993013097-A1 ANTI-RHEUMATIC NAPHTHYRIDINE DERIVATIVES THE BOOTS COMPANY PLC (GB) 1993-07-08 WO disclosed