SCHEMBL8615265

SCHEMBL8615265

CCCCS(=O)(=O)Nc1cccc2nc(-c3ccccc3)cc(NC(=N)NC=O)c12

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MRGPRX1 Q96LB2 1/20 0.37
ACP1 P24666 1/20 0.36
ADORA1 P30542 1/20 0.36
ALDH1A1 P00352 1/20 0.36
THRB P10828 1/20 0.36
HPGD P15428 1/20 0.36
DHODH Q02127 1/20 0.35
ABCB1 P08183 1/20 0.35
ABCC1 P33527 1/20 0.35
ABCG2 Q9UNQ0 1/20 0.35
PGAM1 P18669 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8614953 0.92 ALDH1A1 (0.42) ACP1ADORA1ALDH1A1THRBHPGD
SCHEMBL8615331 0.86 ALDH1A1 (0.41) ACP1ALDH1A1THRBHPGDABCB1
SCHEMBL8620923 0.82 ALOX5AP (0.38)
SCHEMBL8617861 0.82 DHODH (0.42) ACP1ADORA1DHODHABCB1ABCC1
SCHEMBL8613506 0.81 ALDH1A1 (0.45) ALDH1A1THRBHPGD
SCHEMBL8619792 0.81 ADORA1 (0.47) ACP1ADORA1ALDH1A1HPGDABCB1
SCHEMBL8614064 0.80 ABCB1 (0.50) ACP1ADORA1ALDH1A1HPGDABCB1
SCHEMBL8618955 0.79 ACLY (0.41) MRGPRX1ACP1ADORA1ABCB1ABCC1
SCHEMBL8617822 0.79 ACLY (0.38) MRGPRX1ACP1ADORA1DHODHABCB1
SCHEMBL8618937 0.79 PTGER4 (0.46) ACP1ALDH1A1ABCB1ABCC1ABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed