SCHEMBL8625701

SCHEMBL8625701

Cn1c(=O)oc2cc(C(=O)CBr)cnc21

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
HPGD P15428 1/20 0.40
GSK3B P49841 5/20 0.34
KDM4E B2RXH2 1/20 0.33
SIGMAR1 Q99720 2/20 0.32
HSD17B10 Q99714 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
SPR P35270 2/20 0.31
PTPN1 P18031 2/20 0.31
POLB P06746 1/20 0.31
KCNJ1 P48048 2/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8917897 0.87 SIGMAR1 (0.42) ALDH1A1HPGDKDM4ESIGMAR1L3MBTL1
SCHEMBL8626905 0.82 ALDH1A1 (0.43) ALDH1A1HPGDKDM4ESIGMAR1HSD17B10
SCHEMBL8919469 0.82 MAPK1 (0.36) ALDH1A1HPGDSIGMAR1HSD17B10
SCHEMBL8624806 0.80 HSD17B10 (0.35) ALDH1A1HPGDKDM4EHSD17B10L3MBTL1
SCHEMBL8629045 0.79 ALDH1A1 (0.41) ALDH1A1SIGMAR1HSD17B10POLBMEN1
SCHEMBL8919157 0.78 ALDH1A1 (0.35) ALDH1A1HPGDKDM4ESIGMAR1MEN1
SCHEMBL8626022 0.78 ALDH1A1 (0.63) ALDH1A1HPGDKDM4ESIGMAR1HSD17B10
SCHEMBL8625029 0.76 NPC1 (0.48) ALDH1A1HPGDKDM4EHSD17B10L3MBTL1
SCHEMBL8948117 0.74 ALDH1A1 (0.62) ALDH1A1HPGDGSK3BKDM4ESIGMAR1
SCHEMBL7328412 0.74 HSD17B10 (0.53) ALDH1A1HPGDGSK3BKDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5767128-A ANALGESICS ADIR ET COMPAGNIE (FR) 1998-06-16 US disclosed
US-5618819-A ANALGESICS ADIR ET COMPAGNIE (FR) 1997-04-08 US disclosed
EP-0691339-A1 Amine derivatives of 1,3-dihydro-2H-pyrrolo(2,3-b)pyridin-2-ones and oxazolo(4,5-b)pyridin-2(3H)-ones, their process of preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1996-01-10 EP disclosed