SCHEMBL8919157

SCHEMBL8919157

Cn1c(=O)oc2cc(C(=O)CN3CCSCC3)cnc21

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.35
HTT P42858 1/20 0.35
HPGD P15428 1/20 0.34
NOS3 P29474 1/20 0.34
NOS1 P29475 1/20 0.34
NOS2 P35228 1/20 0.34
LMNA P02545 2/20 0.34
SIGMAR1 Q99720 1/20 0.34
KDM4E B2RXH2 2/20 0.33
USP14 P54578 1/20 0.33
NPC1 O15118 1/20 0.33
MAPT P10636 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
GAA P10253 1/20 0.32
ENPP2 Q13822 1/20 0.31
KDM1A O60341 1/20 0.31
MAOA P21397 1/20 0.30
MAOB P27338 1/20 0.30
PDE5A O76074 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8629045 0.87 ALDH1A1 (0.41) ALDH1A1HTTSIGMAR1MAPTMEN1
SCHEMBL8919271 0.82 ALDH1A1 (0.53) ALDH1A1HPGDKDM4EMAPTKMT2A
SCHEMBL8919693 0.82 POLB (0.46) ALDH1A1KDM4EMAPTMEN1KMT2A
SCHEMBL8920278 0.79 MEN1 (0.51) ALDH1A1LMNASIGMAR1NPC1MEN1
SCHEMBL8917897 0.79 SIGMAR1 (0.42) ALDH1A1HPGDLMNASIGMAR1KDM4E
SCHEMBL8625701 0.78 ALDH1A1 (0.40) ALDH1A1HPGDSIGMAR1KDM4EMEN1
SCHEMBL8919198 0.76 POLB (0.47) ALDH1A1LMNAKDM4EMAPTGAA
SCHEMBL8626905 0.75 ALDH1A1 (0.43) ALDH1A1HTTHPGDLMNASIGMAR1
SCHEMBL8919469 0.72 MAPK1 (0.36) ALDH1A1HPGDLMNASIGMAR1
SCHEMBL8921274 0.67 ALDH1A1 (0.45) ALDH1A1KDM4EMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5618819-A ANALGESICS ADIR ET COMPAGNIE (FR) 1997-04-08 US disclosed
EP-0691339-A1 Amine derivatives of 1,3-dihydro-2H-pyrrolo(2,3-b)pyridin-2-ones and oxazolo(4,5-b)pyridin-2(3H)-ones, their process of preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1996-01-10 EP disclosed